Target Details
| UniProt AC | Q04759 |
|---|---|
| Gene Symbol | PRKCQ |
| Protein Name | Protein kinase C theta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 750
- Clinical molecules 360
- Avg pChEMBL 7.71
KEGG Pathways (12)
- Adipocytokine signaling pathway
- Autophagy - animal
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NF-kappa B signaling pathway
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Shigellosis
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Vascular smooth muscle contraction
Active Molecules (750)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TWDPQJRHLMLPRP
|
8.4 | IC50 | 3 | Yes | |
AZHZQWZIQCSEHF
|
8.4 | IC50 | 3 | Yes | |
PPZGIXPLPSHEHY
|
8.4 | IC50 | 2 | — | |
HTLCUINLPKLTDS
|
8.4 | IC50 | 2 | — | |
NIAJEEMQNUPFJB
|
8.4 | IC50 | 3 | Yes | |
NMRUWPRCOQSHGH
|
8.4 | IC50 | 3 | Yes | |
ZQKCTEOSJBBWBB
|
8.4 | IC50 | 3 | Yes | |
KJYFFRNQSIBKHB
|
8.3 | IC50 | 3 | Yes | |
OLTHFAIHFDAJGG
|
8.3 | IC50 | 5 | Yes | |
LDOVNQRBIRULSI
|
8.3 | IC50 | 2 | — | |
IWZNOWDHBWUZLK
|
8.3 | IC50 | 3 | Yes | |
OFAWVNTWBAYIQM
|
8.3 | IC50 | 3 | Yes | |
SSAAQMIJVVUWDZ
|
8.3 | IC50 | 2 | — | |
TUKOILYAIRACKC
|
8.3 | IC50 | 7 | Yes | |
IDSZLHFEKAUIOL
|
8.3 | IC50 | 7 | Yes | |
LIBYFWGPQJFMMW
|
8.3 | IC50 | 2 | Yes | |
TUIMWIXUUASFOT
|
8.3 | IC50 | 2 | — | |
CLAXUCQFRATVEQ
|
8.3 | IC50 | 3 | Yes | |
SJLWKRZGICWCDL
|
8.3 | IC50 | 3 | Yes | |
VKWRGMLRFOFLFQ
|
8.3 | IC50 | 3 | Yes | |
ZKROVQCECIHHES
|
8.3 | IC50 | 3 | Yes | |
AZEVIHVCFXQWCI
|
8.3 | IC50 | 3 | Yes | |
CZYUVYJLWVYZNM
|
8.3 | Ki | 2 | — | |
FNLZNOBAYWDBFQ
|
8.3 | Ki | 2 | — | |
JKLDSNMMVPQIRH
|
8.3 | Ki | 2 | — | |
UVZVWLFSZNPMBS
|
8.3 | IC50 | 17 | — | |
QJVMNACFDUTHPM
|
8.3 | IC50 | 6 | — | |
DHUPFOOXPODTRC
|
8.3 | IC50 | 3 | Yes | |
GAOWZWXUASHKMF
|
8.3 | IC50 | 2 | — | |
GFLGIZVUCFIBRB
|
8.3 | IC50 | 3 | Yes | |
MEAHLUNWZGONEH
|
8.3 | IC50 | 3 | Yes | |
OTBKLEUJZBEEEQ
|
8.3 | IC50 | 3 | Yes | |
XYUFCXJZFZPEJD
|
8.3 | Ki | 23 | Yes | |
BTFQHCKJTLZZRE
|
8.3 | IC50 | 3 | Yes | |
CLENZPTUQALSKC
|
8.3 | IC50 | 3 | Yes | |
OHQBRPBJOMAGLO
|
8.2 | IC50 | 3 | Yes | |
BSPJFZBMQCBCCJ
|
8.2 | IC50 | 3 | Yes | |
OWLWQUHZHTVSAN
|
8.2 | IC50 | 6 | — | |
ZRTHIYZKVPIBMW
|
8.2 | IC50 | 3 | Yes | |
AUQFRAINFQCKDW
|
8.2 | IC50 | 2 | — | |
CEUSLGXUKGZQEI
|
8.2 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
8.2 | IC50 | 408 | — | |
JGWRKYUXBBNENE
|
8.2 | Kd | 11 | — | |
KRSQMQFKFCQXKG
|
8.2 | IC50 | 3 | Yes | |
NGBKJSCBALSPIB
|
8.2 | IC50 | 2 | — | |
SONJXLIPDOXRGA
|
8.2 | IC50 | 3 | Yes | |
WQSBBBAQXNAUEM
|
8.2 | Ki | 2 | — | |
XPKKUXKJOCVNEJ
|
8.2 | IC50 | 3 | Yes | |
JNXDDALKPXMKQB
|
8.2 | IC50 | 3 | Yes | |
KXRUTZLUYFIXDZ
|
8.2 | IC50 | 3 | Yes |