Target Details
| UniProt AC | Q04759 |
|---|---|
| Gene Symbol | PRKCQ |
| Protein Name | Protein kinase C theta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 750
- Clinical molecules 360
- Avg pChEMBL 7.71
KEGG Pathways (12)
- Adipocytokine signaling pathway
- Autophagy - animal
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NF-kappa B signaling pathway
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Shigellosis
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Vascular smooth muscle contraction
Active Molecules (750)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KYJCVYZGCYEQEA
|
8.6 | IC50 | 2 | — | |
VLEXKLPWUMHBQI
|
8.6 | IC50 | 3 | Yes | |
XNMSYXSCPKOHED
|
8.6 | IC50 | 2 | — | |
DGKQFAFCFMHDSZ
|
8.5 | IC50 | 2 | — | |
LPMWTDXPUOFZOV
|
8.5 | Ki | 7 | — | |
NSFBPGFZYOFNAV
|
8.5 | IC50 | 2 | — | |
UJBAYCIQPBHHBB
|
8.5 | IC50 | 3 | Yes | |
USYSUTGHQKSLCI
|
8.5 | IC50 | 3 | Yes | |
UVMAGXADFJGZHF
|
8.5 | IC50 | 2 | — | |
UYBWOWHCXDBQRO
|
8.5 | IC50 | 6 | — | |
ZOLFIIXPYNTFPH
|
8.5 | IC50 | 2 | — | |
AJWYNSXOWAWFRT
|
8.5 | IC50 | 3 | Yes | |
BLWOBXIQFDYTRF
|
8.5 | IC50 | 2 | — | |
FDCMEPRGSNNHNX
|
8.5 | Ki | 4 | — | |
FHISAROGPSYNME
|
8.5 | Ki | 10 | — | |
GJMVLMAOGOJJAE
|
8.5 | IC50 | 2 | — | |
UDPITYZQIVOTOD
|
8.5 | IC50 | 3 | Yes | |
BPPBYLMSKBUXJS
|
8.5 | IC50 | 2 | — | |
CDJHHHAMGANBEP
|
8.5 | IC50 | 2 | — | |
LHQWPYOYDRVMFI
|
8.5 | Ki | 21 | — | |
DAQIKFLEHCFYPH
|
8.5 | IC50 | 3 | Yes | |
CVCIQKJLZNEUAZ
|
8.5 | IC50 | 7 | Yes | |
NHUUGFXCEGPDQR
|
8.5 | IC50 | 2 | — | |
ZWZYAJQDNYIAOM
|
8.5 | IC50 | 2 | — | |
BBBHEOUFBLBBFQ
|
8.5 | IC50 | 2 | — | |
DNZGKSANTHABGF
|
8.5 | IC50 | 3 | Yes | |
GCWARPTUQCJUSX
|
8.5 | IC50 | 3 | Yes | |
PCMKNGBJTSLXPM
|
8.5 | IC50 | 3 | Yes | |
CKAIRTHTMUCHRJ
|
8.4 | IC50 | 2 | — | |
CKQYXXGKHKORSG
|
8.4 | IC50 | 2 | — | |
HFSXGAKDODZJBV
|
8.4 | IC50 | 3 | Yes | |
JVSULVHQOCWQHQ
|
8.4 | IC50 | 3 | Yes | |
OAKTUZHANZGXOY
|
8.4 | IC50 | 2 | — | |
QHJQKYAQVKTFLI
|
8.4 | IC50 | 2 | — | |
UJYYVUFESIJSEY
|
8.4 | IC50 | 3 | Yes | |
XUDDPIKSCLCQKJ
|
8.4 | IC50 | 3 | Yes | |
CRPUDAVZTZIKMJ
|
8.4 | IC50 | 7 | Yes | |
HTPZZARNXXDSIZ
|
8.4 | IC50 | 2 | — | |
JHFLXYPDFJHPMX
|
8.4 | IC50 | 6 | — | |
NSDQNZWGKOYDRS
|
8.4 | IC50 | 2 | — | |
HLTRFCVVQYHUFQ
|
8.4 | IC50 | 2 | — | |
YCLDWGHXCMAHSI
|
8.4 | IC50 | 2 | — | |
BUCGAQTZOOCIRW
|
8.4 | IC50 | 5 | Yes | |
MCQPMCDEXWCMDM
|
8.4 | Ki | 2 | — | |
NWMPVMMGSHXANZ
|
8.4 | Ki | 58 | — | |
QHLWNCNFYOUHJB
|
8.4 | IC50 | 2 | — | |
WQEXBJWFPAMSGJ
|
8.4 | Ki | 8 | Yes | |
XJYBZBREOWBYIA
|
8.4 | IC50 | 3 | Yes | |
ZZMMPNUJLCNYOP
|
8.4 | IC50 | 2 | — | |
ODKAPLPAZCAUMR
|
8.4 | IC50 | 2 | — |