Target Details
| UniProt AC | Q04759 |
|---|---|
| Gene Symbol | PRKCQ |
| Protein Name | Protein kinase C theta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 750
- Clinical molecules 360
- Avg pChEMBL 7.71
KEGG Pathways (12)
- Adipocytokine signaling pathway
- Autophagy - animal
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NF-kappa B signaling pathway
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Shigellosis
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Vascular smooth muscle contraction
Active Molecules (750)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DFRRTVUTEGCPAR
|
8.8 | IC50 | 2 | — | |
HOTMBRBDTHIOMH
|
8.8 | IC50 | 3 | Yes | |
JELDBBFVVGTYRF
|
8.8 | IC50 | 2 | Yes | |
ZCBUQCWBWNUWSU
|
8.8 | Ki | 11 | — | |
ITOPVUHELOTFOX
|
8.8 | IC50 | 3 | Yes | |
NVSJOASGKCGXBZ
|
8.8 | IC50 | 16 | Yes | |
OWWZQKFMHXISPG
|
8.8 | IC50 | 2 | — | |
REZJFFFRLYLHFH
|
8.8 | IC50 | 2 | — | |
KAJIDAUQCMSGGN
|
8.7 | IC50 | 8 | Yes | |
SOEHEJRHIBCBAH
|
8.7 | IC50 | 2 | — | |
WJNGWUFYYQTNGU
|
8.7 | IC50 | 2 | — | |
JYQVFPCZFZOPCW
|
8.7 | IC50 | 2 | — | |
OZTYUUKHFRSKCQ
|
8.7 | IC50 | 2 | — | |
PBWBADGNVJJHFC
|
8.7 | IC50 | 3 | Yes | |
BYDKAYRDAFQMFD
|
8.7 | IC50 | 2 | — | |
CDSMPVVXLHABBR
|
8.7 | IC50 | 2 | — | |
FEFAAFLIBQXOAO
|
8.7 | IC50 | 2 | — | |
GLKZLGGCNUQEAN
|
8.7 | IC50 | 3 | Yes | |
HKSZLNNOFSGOKW
|
8.7 | Ki | 118 | — | |
IDMUMGBXJGYJTD
|
8.7 | Ki | 3 | — | |
JKLDSNMMVPQIRH
|
8.7 | Ki | 2 | — | |
ORIFTCPILCBZCQ
|
8.7 | IC50 | 2 | — | |
QYBVZIIWBRIXMX
|
8.7 | IC50 | 12 | Yes | |
ZNFICDKPLIEJJT
|
8.7 | IC50 | 2 | — | |
AAKDVUMRVXYBST
|
8.7 | IC50 | 2 | — | |
CIVFNZIOXQANAM
|
8.7 | IC50 | 5 | — | |
KMFOKKGKNMQAAN
|
8.7 | IC50 | 6 | — | |
LBKFIWNOGYSLHE
|
8.7 | IC50 | 2 | — | |
OXPLGRNOXPCLEB
|
8.7 | IC50 | 3 | Yes | |
TUJXMCOKEYNEHL
|
8.7 | IC50 | 2 | — | |
UPSXKHFTVWTQRJ
|
8.7 | IC50 | 2 | — | |
YIAUOBNZXMZCFP
|
8.7 | IC50 | 2 | — | |
COOZRRUJSWPFHC
|
8.7 | IC50 | 3 | Yes | |
JZLFYMHIISZQCZ
|
8.7 | IC50 | 12 | Yes | |
LOOCBXNRYHTANC
|
8.7 | IC50 | 2 | — | |
LTFWFNLDCHAVQF
|
8.7 | IC50 | 2 | — | |
SUKUYCBPKLCSMU
|
8.7 | IC50 | 2 | — | |
IWPNPNGPAZFVCZ
|
8.6 | IC50 | 3 | Yes | |
HDYPWSDXJZTYPP
|
8.6 | IC50 | 3 | Yes | |
UVUMDKAWNBACHR
|
8.6 | IC50 | 3 | Yes | |
YTAXZQBKZAMFER
|
8.6 | IC50 | 3 | Yes | |
ZCBUQCWBWNUWSU
|
8.6 | Kd | 59 | — | |
ZDISSWUDAVTQSK
|
8.6 | IC50 | 3 | Yes | |
YPXYBPVNHTYOHY
|
8.6 | IC50 | 2 | — | |
YQOOLLWMVHTWOY
|
8.6 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
8.6 | Kd | 599 | — | |
UZDDRLFGKXVQQG
|
8.6 | IC50 | 2 | — | |
WNEWTOQENXHIHL
|
8.6 | IC50 | 2 | — | |
HEUDUTKTUQTOGI
|
8.6 | IC50 | 2 | — | |
IFLKFPIAJMOXTG
|
8.6 | IC50 | 3 | Yes |