Target Details
| UniProt AC | Q04759 |
|---|---|
| Gene Symbol | PRKCQ |
| Protein Name | Protein kinase C theta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 750
- Clinical molecules 360
- Avg pChEMBL 7.71
KEGG Pathways (12)
- Adipocytokine signaling pathway
- Autophagy - animal
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NF-kappa B signaling pathway
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Shigellosis
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Vascular smooth muscle contraction
Active Molecules (750)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VWMGVMIQUFQRRV
|
9.1 | IC50 | 2 | — | |
WDARYLSSWBWVCU
|
9.1 | Ki | 49 | — | |
YTUIPBJVDYRJDG
|
9.1 | IC50 | 2 | — | |
ICQQDVZUHPTFPS
|
9.1 | IC50 | 3 | Yes | |
LLMXWBSEQIDLJG
|
9.1 | IC50 | 5 | — | |
AXXPOMJMORIBKL
|
9.1 | IC50 | 2 | — | |
TVJVIPXZACZIIC
|
9.1 | IC50 | 2 | — | |
OLYCNNWWUIENNA
|
9.1 | IC50 | 2 | — | |
SZJIXBKHTOPEKG
|
9.1 | IC50 | 6 | Yes | |
VHOMUDQDZZWLSZ
|
9.1 | IC50 | 3 | — | |
MFDKBLCTDGSTAK
|
9.1 | IC50 | 2 | — | |
HXWARSZQGAFXJM
|
9.0 | IC50 | 7 | — | |
VZTQRSJQRWBYFW
|
9.0 | IC50 | 2 | — | |
KQKVTOFNZCMSEP
|
9.0 | IC50 | 2 | — | |
OAVGBZOFDPFGPJ
|
9.0 | IC50 | 42 | Yes | |
PDSONWYECZHBAE
|
9.0 | Ki | 2 | — | |
PDSONWYECZHBAE
|
9.0 | IC50 | 3 | — | |
RDFXBYJUHGEYHA
|
9.0 | IC50 | 9 | Yes | |
SKUHDUHJJACTNK
|
9.0 | IC50 | 2 | — | |
FPSGCBWWRUZTIV
|
8.9 | IC50 | 3 | Yes | |
MZHAAXPSUZZVJO
|
8.9 | IC50 | 2 | — | |
NQESDTBKBPAEPS
|
8.9 | IC50 | 2 | — | |
REGYZNVOEPVCIC
|
8.9 | IC50 | 2 | — | |
SUKUYCBPKLCSMU
|
8.9 | IC50 | 2 | — | |
URLJNGHIJZMXTK
|
8.9 | IC50 | 6 | — | |
UZGZCPNOEILBMK
|
8.9 | IC50 | 2 | — | |
ZOLWRJUQMXEKEO
|
8.9 | IC50 | 6 | — | |
ATTAVUMAVKBGLW
|
8.9 | IC50 | 3 | Yes | |
DKGIQYXYEVWNNO
|
8.9 | IC50 | 2 | — | |
DNZGKSANTHABGF
|
8.9 | IC50 | 3 | Yes | |
FEFPSHIDVWKVSO
|
8.9 | IC50 | 4 | — | |
ISHUULBGXOVLLF
|
8.9 | IC50 | 2 | — | |
LPLRIFJSFFHUQM
|
8.9 | IC50 | 3 | — | |
NPIKPVAKTCZWAG
|
8.9 | IC50 | 2 | — | |
RKEQTICDODWVQT
|
8.9 | IC50 | 2 | — | |
RRGJUOHIDUNWCQ
|
8.9 | IC50 | 2 | — | |
SNIZLDGVUOKDEA
|
8.9 | IC50 | 3 | Yes | |
XEHZTUCPROUDNJ
|
8.9 | IC50 | 3 | Yes | |
DASVAQCTVIQROX
|
8.8 | Ki | 8 | Yes | |
JMBOYLIMLIXSDW
|
8.8 | IC50 | 3 | Yes | |
NLJJDZMBYLCWHR
|
8.8 | IC50 | 2 | — | |
QZIHHXYMIRLTTO
|
8.8 | IC50 | 3 | Yes | |
CFGWNLDQFLAEHP
|
8.8 | IC50 | 2 | — | |
FVAXCXHKGMJCLC
|
8.8 | IC50 | 4 | — | |
JPINQKLMVKTGTL
|
8.8 | IC50 | 3 | Yes | |
MMFFLYVAVCPQHO
|
8.8 | IC50 | 3 | Yes | |
VEKVVEWREDUQML
|
8.8 | IC50 | 2 | — | |
WALDOGJQTYJBFG
|
8.8 | IC50 | 3 | Yes | |
WFUUKKJTZMFANX
|
8.8 | IC50 | 2 | — | |
XYKVGXVSUAFNLB
|
8.8 | IC50 | 3 | Yes |