Target Details
| UniProt AC | Q04759 |
|---|---|
| Gene Symbol | PRKCQ |
| Protein Name | Protein kinase C theta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 750
- Clinical molecules 360
- Avg pChEMBL 7.71
KEGG Pathways (12)
- Adipocytokine signaling pathway
- Autophagy - animal
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NF-kappa B signaling pathway
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Shigellosis
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Vascular smooth muscle contraction
Active Molecules (750)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DCHKISSMZIQZRF
|
7.4 | IC50 | 2 | — | |
KEBDGBLZUWTDQL
|
7.4 | IC50 | 3 | Yes | |
RCKVYOXLMHAPMO
|
7.4 | IC50 | 3 | Yes | |
IJYPXTWDRNLKMU
|
7.4 | IC50 | 3 | Yes | |
CNXKJMKQJSETCG
|
7.4 | IC50 | 3 | — | |
DKXHSOUZPMHNIZ
|
7.4 | Ki | 51 | Yes | |
KJGUOQMSLKZPAT
|
7.4 | IC50 | 17 | Yes | |
GHCPXYAHSHXFSC
|
7.4 | IC50 | 3 | Yes | |
HAWYDMHDXJUGRR
|
7.4 | IC50 | 3 | Yes | |
NTUVEMUMVHHACY
|
7.4 | IC50 | 12 | Yes | |
JMRDOCPDIXFWLY
|
7.4 | IC50 | 3 | Yes | |
OGFRRHMGGJQLRU
|
7.4 | IC50 | 3 | Yes | |
HHLNVCKLKSYSJN
|
7.4 | IC50 | 3 | Yes | |
VDBJPTBJJMQNOW
|
7.4 | IC50 | 6 | — | |
WKZTVBCDQYBGBO
|
7.3 | IC50 | 16 | Yes | |
GDORNNADINCMRQ
|
7.3 | IC50 | 2 | Yes | |
RQFQHXQYIYDKMC
|
7.3 | IC50 | 3 | Yes | |
AYCPARAPKDAOEN
|
7.3 | IC50 | 73 | — | |
DOCCMHSNEKDEOV
|
7.3 | IC50 | 3 | Yes | |
MDHNNGDJYHAYKJ
|
7.3 | IC50 | 12 | Yes | |
QQTVBLADGKPBRJ
|
7.3 | Ki | 2 | — | |
CYRPAUWSHGGREB
|
7.3 | Ki | 8 | Yes | |
MWKQDYOZWRAWMS
|
7.3 | IC50 | 3 | Yes | |
OJCFURIPWIIKNL
|
7.3 | IC50 | 2 | — | |
OVELCOBTBDZAMT
|
7.3 | IC50 | 2 | Yes | |
OAKNYDVXYJXOEP
|
7.3 | IC50 | 2 | Yes | |
QEPARSUKSLKMMO
|
7.3 | IC50 | 7 | Yes | |
VKLQFIYLAKBNIW
|
7.3 | IC50 | 3 | Yes | |
HUWJTNZRWNYRJP
|
7.3 | IC50 | 2 | — | |
UHVOJNPWRWKQSP
|
7.3 | IC50 | 3 | Yes | |
YUJAAMQBNNAQRP
|
7.3 | IC50 | 6 | — | |
KVPCAWMJGFMDHN
|
7.2 | IC50 | 3 | Yes | |
AAFUKFIIJDVJOX
|
7.2 | IC50 | 2 | — | |
DEUHHHBUOZFXCN
|
7.2 | IC50 | 3 | Yes | |
MPKJLCGWZCOAHC
|
7.2 | IC50 | 3 | Yes | |
ORSMLITYQOYOSE
|
7.2 | IC50 | 2 | — | |
XOIXULDEDZVLBV
|
7.2 | IC50 | 2 | — | |
AFICENYJQYURCA
|
7.2 | Ki | 2 | — | |
DBENCPRFMOMLTO
|
7.2 | IC50 | 2 | — | |
OQICVMYHDNIADM
|
7.2 | IC50 | 6 | — | |
LBFYQISQYCGDDW
|
7.2 | Ki | 7 | — | |
LURPXFLMWSMKCY
|
7.2 | Ki | 2 | — | |
MVQGUYKZTHVOEH
|
7.2 | Ki | 8 | Yes | |
RVIJQMOQZFCSHL
|
7.2 | Ki | 8 | Yes | |
XXIWRTOLXWAEJC
|
7.2 | IC50 | 13 | Yes | |
MLGGUGPIWDHBAI
|
7.2 | Ki | 33 | — | |
OQCCQWBVUGOVBA
|
7.2 | Ki | 2 | — | |
OWRXHGAFWZFFCW
|
7.2 | Ki | 113 | — | |
RKUKAACYUCUJEE
|
7.2 | Ki | 58 | — | |
TUBBFDZWFNUZLH
|
7.2 | IC50 | 12 | Yes |