Target Details
| UniProt AC | Q04759 |
|---|---|
| Gene Symbol | PRKCQ |
| Protein Name | Protein kinase C theta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 750
- Clinical molecules 360
- Avg pChEMBL 7.71
KEGG Pathways (12)
- Adipocytokine signaling pathway
- Autophagy - animal
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NF-kappa B signaling pathway
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Shigellosis
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Vascular smooth muscle contraction
Active Molecules (750)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WTXAWDOYPWWUJL
|
10.1 | IC50 | 11 | — | |
FANQQVWXAKUWNI
|
10.0 | IC50 | 6 | — | |
REAZZDPREXHWNV
|
10.0 | Ki | 7 | — | |
SSXCVTWCXHGTLK
|
9.9 | IC50 | 11 | — | |
WESMIFKYYUDSHE
|
9.9 | IC50 | 2 | — | |
XFQSFVPULNZYER
|
9.9 | IC50 | 2 | — | |
KTGVSZYYHHRRGW
|
9.8 | IC50 | 11 | — | |
VIESIZQAHOPEBR
|
9.8 | IC50 | 11 | — | |
LJCBQNDNKZTPPD
|
9.8 | IC50 | 2 | — | |
RHJPBGWFGOAEID
|
9.8 | Ki | 8 | Yes | |
NVYBXIDWOJVGQI
|
9.8 | IC50 | 11 | — | |
APVOCXHEVZBCGS
|
9.7 | IC50 | 11 | — | |
VJMOXJYFZUYUTA
|
9.7 | IC50 | 2 | — | |
XSJFPSCYMJFDNI
|
9.7 | Ki | 7 | — | |
DHTLXMRCLSUJPP
|
9.7 | IC50 | 11 | — | |
CCFSCBCNTYCQQD
|
9.6 | IC50 | 4 | — | |
NJDCTLINWXDFST
|
9.6 | IC50 | 2 | — | |
JWHUZKCDLIXMSE
|
9.6 | IC50 | 4 | — | |
PPSTZDPKWJXFIH
|
9.6 | IC50 | 2 | — | |
VHLRDCSSMVVRQX
|
9.6 | IC50 | 2 | — | |
DZIUPOCVDSYPSY
|
9.6 | IC50 | 8 | Yes | |
IUQRWIKPYXRDAP
|
9.5 | IC50 | 2 | — | |
DWUYMGRQDSNZNZ
|
9.5 | IC50 | 2 | — | |
ZWFTUJOJJZSCMP
|
9.5 | IC50 | 2 | — | |
KNTODVAJZPLTBO
|
9.5 | IC50 | 4 | — | |
ZYKISFVIHSEGIE
|
9.5 | IC50 | 2 | — | |
AODINEOJAWVRMB
|
9.4 | IC50 | 2 | — | |
VVRRZOFLLJAMIK
|
9.4 | IC50 | 11 | — | |
YNARAQPWBNWRIS
|
9.4 | IC50 | 3 | — | |
XXJXHXJWQSCNPX
|
9.4 | IC50 | 7 | — | |
DFHNPLPBHYMUAW
|
9.4 | IC50 | 2 | — | |
KRMLZRDHQHQPJW
|
9.4 | IC50 | 5 | Yes | |
SDEAUNNPTULCST
|
9.3 | IC50 | 3 | — | |
UJKQZOOHKSDLBL
|
9.3 | IC50 | 2 | — | |
GXRHJQDLOAPBIK
|
9.3 | IC50 | 3 | Yes | |
GMQQMSKNSNVPOW
|
9.3 | IC50 | 9 | Yes | |
WAKGEHXTOOFEAE
|
9.3 | IC50 | 27 | — | |
SWKUTOXEFLDOID
|
9.3 | Ki | 7 | — | |
CMIRYEYYRRGPKG
|
9.2 | IC50 | 3 | — | |
UZCZCOMLMMSRLY
|
9.2 | IC50 | 6 | — | |
CDVWLKDMFLAJTO
|
9.2 | IC50 | 2 | — | |
FBYHLMJXXHAYDR
|
9.2 | IC50 | 2 | — | |
WUJFWMRQXPIJIN
|
9.2 | IC50 | 3 | Yes | |
MKCCHIFQLCHEBR
|
9.2 | IC50 | 3 | Yes | |
PBMUEOYWGJZICW
|
9.2 | IC50 | 4 | — | |
ZVWUCVHEPQALQU
|
9.2 | IC50 | 2 | — | |
WPDAGVJJKLBFOI
|
9.2 | IC50 | 2 | — | |
MNLOLQHZWGLJBO
|
9.2 | IC50 | 2 | — | |
BQJRUJTZSGYBEZ
|
9.1 | Kd | 13 | Yes | |
QZCYXWFWSDBJGL
|
9.1 | Ki | 8 | Yes |