Target Details
UniProt ACQ04756
Gene SymbolHGFAC
Protein NameHepatocyte growth factor activator serine protease
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00008 (EGF) PF00040 (fn2) PF00051 (Kringle) PF00089 (Trypsin)
Summary
  • Multi-target molecules 47
  • Clinical molecules 1
  • Avg pChEMBL 7.1
Top Co-occurrence Targets
Active Molecules (47)
InChIKey pChEMBL Type Targets Clinical
SVOXYTTZYOSESO 8.4 Ki 4
ZLIIZOMJAUACIT 8.3 IC50 4
MMCZPBUBUPXIQM 8.1 Ki 4
DIOWGKUHSWDAQR 7.9 Ki 3
RJBLHAMXODQZMM 7.9 IC50 4
CNVNITMLGKDQQY 7.8 Ki 3
WKFXBFMYZUNDEO 7.7 Ki 3
DVZQOTUGXDAQNJ 7.6 Ki 3
MQQNFDZXWVTQEH 7.6 Ki 11
QQRQFIXRVWJLNT 7.6 Ki 10
MDTKEYLCTKYBSK 7.6 IC50 4
NEQGCINBAXAQKD 7.6 IC50 5
WQISNVQCRKRHME 7.5 Ki 4
AIAPZNJOJFJSQR 7.5 IC50 4
BLOFNYQHKSGSGE 7.5 Ki 3
ZTZVSJUJOHEBFJ 7.4 IC50 4
PFSNIQDNVQKULM 7.3 Ki 3
UNOVDKDICJRWRT 7.2 Ki 3
CFSDWWHMXFUPKB 7.2 Ki 3
GWIRLHLNQLEUAV 7.2 Ki 3
RETMNWIAJUVWLF 7.2 Ki 3
GBWLZSRRLJETHI 7.2 IC50 5
PHPJWSFXNNRMES 7.2 Ki 3
BSCYVKJQDUSMFJ 7.2 Ki 3
KJLKBVQGEXTILS 7.1 Ki 3
ZRJSFZXXCBTZHR 7.1 Ki 3
AGLYIVQPVAYVMN 7.1 Ki 3
AIAPZNJOJFJSQR 7.1 IC50 4
QNGSZDJLWYVTQN 7.0 Ki 3
VFNBZASFQVJNJZ 7.0 Ki 3
QYGNVWAMIWRSDZ 6.8 Ki 7
LNFLFMVSXZPRHU 6.7 Ki 3
GDBQQVLCIARPGH 6.7 Ki 10
OLNJKAXRBXUBTB 6.7 Ki 10 Yes
YNTWFQFGHYXDEM 6.6 Ki 7
PLLBBBICXMICNE 6.6 IC50 4
QCZLVVCFUACPGA 6.5 Ki 3
PDYWNBXTWVNQDC 6.5 Ki 7
BFOHAEDJCBXVHR 6.4 Ki 5
SNXRYLUCKVDDCE 6.4 Ki 7
GBFNBYMSXRCRBZ 6.4 Ki 7
MBBPFTAWIJCEBL 6.3 Ki 3
HGBLIBDRBSWLRN 6.3 Ki 7
FMYZVNGLLMHTNV 6.3 Ki 7
CWPABYGTEGMLDD 6.1 IC50 3
HINXTEQWTTZJOH 6.1 Ki 7
XODXDNXIWIHPLC 6.0 Ki 3
2D structure