Target Details
| UniProt AC | Q04609 |
|---|---|
| Gene Symbol | FOLH1 |
| Protein Name | Glutamate carboxypeptidase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02225 (PA) PF04389 (Peptidase_M28) PF04253 (TFR_dimer) |
Summary
- Multi-target molecules 23
- Clinical molecules 0
- Avg pChEMBL 7.86
KEGG Pathways (5)
Active Molecules (23)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ROXRILBFJQYPNZ
|
11.0 | Ki | 2 | — | |
ISEYJGQFXSTPMQ
|
9.5 | IC50 | 2 | — | |
ISEYJGQFXSTPMQ
|
9.4 | IC50 | 2 | — | |
UHUQCJJQRNMUJJ
|
8.7 | IC50 | 2 | — | |
ZUEXRXMHJQFNSG
|
8.7 | IC50 | 3 | — | |
BLTYWXMDJBDQPE
|
8.2 | IC50 | 2 | — | |
SOAPXKSPJAZNGO
|
8.1 | Ki | 2 | — | |
OZXNUTGMCCPZLB
|
8.1 | IC50 | 2 | — | |
PCHRROMHSFRTIA
|
8.0 | IC50 | 2 | — | |
ZUEBVBPVXLQMQR
|
8.0 | Ki | 2 | — | |
QUTRTBDFCYIXBN
|
7.9 | IC50 | 2 | — | |
JIGUYYXQAKEPKB
|
7.8 | IC50 | 2 | — | |
FYBZEJITZIQBMD
|
7.6 | IC50 | 2 | — | |
WMSBVXZOWAWWPP
|
7.6 | Kd | 2 | — | |
VZMSNDLDHMJHAH
|
7.4 | IC50 | 3 | — | |
NEUOTELYJPSZFF
|
7.4 | IC50 | 3 | — | |
DGIMSGNEZGNIDP
|
7.3 | Kd | 2 | — | |
FPNJXNKGPWSIAM
|
7.1 | IC50 | 2 | — | |
WKJXCVSDKZAOAI
|
6.8 | Kd | 2 | — | |
LFOMVPSUFXNQKT
|
6.6 | Kd | 2 | — | |
YNENWAKWCIYFOE
|
6.6 | IC50 | 2 | — | |
IBQPJYGLSNFRAF
|
6.5 | Kd | 2 | — | |
YHAZITYYCGMBQX
|
6.5 | Kd | 2 | — |