Target Details
| UniProt AC | Q03164 |
|---|---|
| Gene Symbol | KMT2A |
| Protein Name | Histone-lysine N-methyltransferase 2A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05965 (FYRC) PF05964 (FYRN) PF00628 (PHD) PF00856 (SET) PF02008 (zf-CXXC) PF13771 (zf-HC5HC2H) |
Summary
- Multi-target molecules 252
- Clinical molecules 0
- Avg pChEMBL 7.03
KEGG Pathways (4)
Associated Diseases (3)
Active Molecules (252)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RRQBQDOLKJVCNU
|
6.0 | IC50 | 2 | — | |
ZXNZFLDTEWCDMC
|
6.0 | IC50 | 2 | — |