Target Details
| UniProt AC | Q03164 |
|---|---|
| Gene Symbol | KMT2A |
| Protein Name | Histone-lysine N-methyltransferase 2A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05965 (FYRC) PF05964 (FYRN) PF00628 (PHD) PF00856 (SET) PF02008 (zf-CXXC) PF13771 (zf-HC5HC2H) |
Summary
- Multi-target molecules 252
- Clinical molecules 0
- Avg pChEMBL 7.03
KEGG Pathways (4)
Associated Diseases (3)
Active Molecules (252)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SUXNCBRCYTZFPW
|
6.3 | IC50 | 5 | — | |
YAYXNECXQXPQIJ
|
6.3 | IC50 | 2 | — | |
CDBKROHOJVKZNJ
|
6.3 | IC50 | 2 | — | |
ZFMZWYQYVCPKDJ
|
6.3 | IC50 | 2 | — | |
IAEZONCHIHJVKX
|
6.3 | IC50 | 2 | — | |
ZAIPJVQTYUSDTG
|
6.3 | IC50 | 5 | — | |
YREYEVIYCVEVJK
|
6.3 | IC50 | 6 | — | |
ZNYQTNBVCYYXDE
|
6.3 | IC50 | 2 | — | |
FWQWFEHDDXOZTR
|
6.3 | IC50 | 2 | — | |
VJMSEJCFUWKXQR
|
6.3 | IC50 | 2 | — | |
XOODMKHLHHLZMP
|
6.3 | IC50 | 2 | — | |
YPMLDLHIIBLGQJ
|
6.3 | IC50 | 2 | — | |
CLIGIUJNVZBOLZ
|
6.3 | IC50 | 2 | — | |
XACXGFXQIQGLQP
|
6.2 | IC50 | 2 | — | |
LCHGERIHAPDZCU
|
6.2 | IC50 | 2 | — | |
ORDFLTLXLXTYCX
|
6.2 | IC50 | 2 | — | |
RPXXFSOUEYJZLT
|
6.2 | IC50 | 5 | — | |
LSSYDYCCKSSRBW
|
6.2 | IC50 | 2 | — | |
PWIXTNXPOYAMKW
|
6.2 | IC50 | 2 | — | |
AVGRXABHJJNRNY
|
6.2 | IC50 | 2 | — | |
FKUKOLIMTPBZQB
|
6.2 | IC50 | 2 | — | |
NJYSIUZZZYJDMM
|
6.2 | IC50 | 2 | — | |
TWQRKOGYUAIFNA
|
6.2 | IC50 | 2 | — | |
CALOBSGMDWBFKP
|
6.2 | IC50 | 2 | — | |
OOOIIBPVHFSXRR
|
6.2 | IC50 | 2 | — | |
ZXGUOQGZIKIBCM
|
6.2 | IC50 | 2 | — | |
WURJOCVDSUSNBQ
|
6.2 | IC50 | 2 | — | |
YPXKTWOWTNYSBN
|
6.2 | IC50 | 2 | — | |
ZJUKTBDSGOFHSH
|
6.1 | IC50 | 22 | — | |
CMZXXROIVBWQKJ
|
6.1 | IC50 | 5 | — | |
CONURMHQMUEEDI
|
6.1 | IC50 | 2 | — | |
DGHMWFXLUQFCNT
|
6.1 | IC50 | 2 | — | |
UWDXJOIFTJGVGJ
|
6.1 | IC50 | 2 | — | |
DFLZGJORZOLMPP
|
6.1 | IC50 | 2 | — | |
DXVHKVAAZWOGEQ
|
6.1 | IC50 | 2 | — | |
FGWGLQMPNQASED
|
6.1 | IC50 | 2 | — | |
FUUKXIVVPBOGQX
|
6.1 | IC50 | 2 | — | |
IAEZONCHIHJVKX
|
6.1 | IC50 | 2 | — | |
LXONEMNSYOAQJT
|
6.1 | IC50 | 2 | — | |
MZXQOJPMACYONE
|
6.1 | IC50 | 2 | — | |
ZHYKLPAWOLFHNY
|
6.1 | IC50 | 2 | — | |
IDXURNUKWGSUOE
|
6.1 | IC50 | 2 | — | |
UDQQSVJQUIZVFV
|
6.1 | IC50 | 2 | — | |
QNXFOPYFFZOHCX
|
6.1 | IC50 | 2 | — | |
RWMJXLQEZZOCBN
|
6.0 | IC50 | 2 | — | |
XXBPCORNASWFLI
|
6.0 | IC50 | 2 | — | |
HJPMPWYSTRBBLP
|
6.0 | IC50 | 2 | — | |
YOZWQAYOZCWKIG
|
6.0 | IC50 | 2 | — | |
HUCHWMVKXDSHCR
|
6.0 | IC50 | 2 | — | |
NDPACLRAEMRBOG
|
6.0 | IC50 | 2 | — |