Target Details
| UniProt AC | Q03164 |
|---|---|
| Gene Symbol | KMT2A |
| Protein Name | Histone-lysine N-methyltransferase 2A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05965 (FYRC) PF05964 (FYRN) PF00628 (PHD) PF00856 (SET) PF02008 (zf-CXXC) PF13771 (zf-HC5HC2H) |
Summary
- Multi-target molecules 252
- Clinical molecules 0
- Avg pChEMBL 7.03
KEGG Pathways (4)
Associated Diseases (3)
Active Molecules (252)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FTSMDZBUBLYVKI
|
6.7 | IC50 | 2 | — | |
GERBHAWOLATBEK
|
6.7 | IC50 | 2 | — | |
JWPMQFAQNDYLNU
|
6.7 | IC50 | 2 | — | |
QTSKXZZDLJLJLM
|
6.7 | IC50 | 5 | — | |
OYQKINJAVGKCOA
|
6.7 | IC50 | 2 | — | |
HYLJRWUMYPYWOV
|
6.7 | IC50 | 2 | — | |
DHBHJVJPRVYFCA
|
6.7 | IC50 | 5 | — | |
QFPZYAHHNKMSAE
|
6.7 | IC50 | 2 | — | |
SYLSWCJVGKVJRP
|
6.7 | IC50 | 2 | — | |
UJCBRBGSYIDHKB
|
6.7 | IC50 | 2 | — | |
ATCFHABJGDDNHA
|
6.7 | IC50 | 2 | — | |
BNDCSLSPYZRORX
|
6.7 | IC50 | 2 | — | |
MPNUDPQVRXYIJO
|
6.7 | IC50 | 2 | — | |
DJOVLOYCGXNVPI
|
6.7 | IC50 | 2 | — | |
DRGVYVUPPVUATJ
|
6.7 | IC50 | 2 | — | |
HVPTXLPRWAIOFE
|
6.6 | IC50 | 2 | — | |
RNNUHFXCYYPDIF
|
6.6 | IC50 | 5 | — | |
FXLINUKVODZXEA
|
6.6 | IC50 | 2 | — | |
INLKZOGWBUSMOY
|
6.6 | IC50 | 2 | — | |
DFMXVFSCNICRHG
|
6.6 | IC50 | 2 | — | |
KAHJAGWFBUHJQJ
|
6.6 | IC50 | 2 | — | |
PHEZBZSOCLLNEW
|
6.6 | IC50 | 2 | — | |
NQNUBXZOPJLVNJ
|
6.6 | IC50 | 2 | — | |
OMMVXYNQHWMPMT
|
6.6 | IC50 | 2 | — | |
ZIWKHOHCZXDNQD
|
6.6 | IC50 | 2 | — | |
PVWSGHIMLSOZLF
|
6.5 | IC50 | 2 | — | |
ADRMGNQFAFGBJJ
|
6.5 | IC50 | 2 | — | |
GOJNJTYVCAMOML
|
6.5 | IC50 | 2 | — | |
YFITWOOGOWMDIU
|
6.5 | IC50 | 2 | — | |
YFITWOOGOWMDIU
|
6.5 | IC50 | 2 | — | |
CXFJNJZPBYIKCK
|
6.5 | IC50 | 2 | — | |
CZWZZEUKNASAHM
|
6.5 | IC50 | 4 | — | |
AKYZOYQVCPKNMI
|
6.5 | IC50 | 2 | — | |
INJQLGJLXFFEBE
|
6.5 | IC50 | 2 | — | |
QNEXYXLSJZBQJZ
|
6.5 | IC50 | 2 | — | |
SILRGLDFBXVGOQ
|
6.5 | IC50 | 5 | — | |
GLHJOTVYVUCLQO
|
6.5 | IC50 | 2 | — | |
UPIPNZWTALWOSN
|
6.5 | IC50 | 2 | — | |
NLPDQBANAXKJTJ
|
6.5 | IC50 | 2 | — | |
SZQUBMQVFOLNKK
|
6.4 | IC50 | 2 | — | |
BFFCPQIDLRDLAH
|
6.4 | IC50 | 2 | — | |
GMHYNYVINHPZGO
|
6.4 | IC50 | 2 | — | |
QBITUTDDFZQXDO
|
6.4 | IC50 | 2 | — | |
RZKSQRIPRKWVBU
|
6.4 | IC50 | 4 | — | |
VVBLYRNNBHAYNU
|
6.4 | IC50 | 2 | — | |
GFXGFUJVRDJZFM
|
6.4 | IC50 | 2 | — | |
OAOHJPWUVQFOCX
|
6.4 | IC50 | 2 | — | |
JZOSRTPOYRYTRA
|
6.3 | IC50 | 5 | — | |
SRQYLNYQAPCPIR
|
6.3 | IC50 | 2 | — | |
DLNBITDSKNXQMK
|
6.3 | IC50 | 2 | — |