Target Details
| UniProt AC | Q03164 |
|---|---|
| Gene Symbol | KMT2A |
| Protein Name | Histone-lysine N-methyltransferase 2A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05965 (FYRC) PF05964 (FYRN) PF00628 (PHD) PF00856 (SET) PF02008 (zf-CXXC) PF13771 (zf-HC5HC2H) |
Summary
- Multi-target molecules 252
- Clinical molecules 0
- Avg pChEMBL 7.03
KEGG Pathways (4)
Associated Diseases (3)
Active Molecules (252)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NPFRAPJTDVLBBW
|
7.1 | IC50 | 5 | — | |
QCTQIUVBBPESJQ
|
7.1 | IC50 | 2 | — | |
QDYDQJXQYYYAHD
|
7.1 | IC50 | 2 | — | |
FQHLCCRHERJGGU
|
7.1 | IC50 | 2 | — | |
UBUIDPURYFKDTJ
|
7.1 | IC50 | 2 | — | |
PRAJCBYVBKZLED
|
7.1 | IC50 | 5 | — | |
TWLPSDLPEQAIFC
|
7.1 | IC50 | 2 | — | |
HOWWOQQFNUIEDX
|
7.0 | IC50 | 2 | — | |
PAQXRXLELGMMTP
|
7.0 | IC50 | 2 | — | |
GPUCGUREPBUUPX
|
7.0 | IC50 | 2 | — | |
WXYILIFTWPRGQC
|
7.0 | IC50 | 2 | — | |
KUBSRASLWYNRKJ
|
7.0 | IC50 | 2 | — | |
TVPHEUCQQXAPKZ
|
7.0 | IC50 | 2 | — | |
XCVJSTZYHUNTCU
|
7.0 | IC50 | 5 | — | |
XIJLQIRAWOEATH
|
7.0 | IC50 | 2 | — | |
ZIWKHOHCZXDNQD
|
7.0 | IC50 | 2 | — | |
FDPSNDOCRPXFCD
|
7.0 | IC50 | 2 | — | |
FNQRCLCAWMTHIP
|
7.0 | IC50 | 2 | — | |
GRCIWJRXZFZJCZ
|
7.0 | IC50 | 2 | — | |
GBEYGHHOGZXQCC
|
7.0 | IC50 | 2 | — | |
NQXVDDGKDJESCO
|
6.9 | IC50 | 2 | — | |
AMSVGXDFPHGXFJ
|
6.9 | IC50 | 5 | — | |
GIWCILLVZIEDKV
|
6.9 | IC50 | 2 | — | |
KXYGAIVJVQJFDQ
|
6.9 | IC50 | 5 | — | |
QDJNCNNOOZJAPQ
|
6.9 | IC50 | 2 | — | |
ZZVXSOZWKGNLLE
|
6.9 | IC50 | 2 | — | |
MWWRLWPCGQFTIQ
|
6.9 | IC50 | 5 | — | |
FDLXLYIFHPVTGM
|
6.9 | IC50 | 2 | — | |
OXSOFPMSKVUQBE
|
6.9 | IC50 | 5 | — | |
VCGGKAFSZXGDJK
|
6.9 | IC50 | 2 | — | |
JGIIYJOEBDGPQO
|
6.9 | IC50 | 5 | — | |
VHPRRJZGFMSHQV
|
6.9 | IC50 | 5 | — | |
PRFGRQZQIVZYDV
|
6.8 | IC50 | 2 | — | |
ZXKYRAQRTUGVRY
|
6.8 | IC50 | 2 | — | |
XNLFOGWQUFHWMA
|
6.8 | IC50 | 2 | — | |
BVTRNKNKLBXNOU
|
6.8 | IC50 | 2 | — | |
UWACKSCSSLOEGH
|
6.8 | IC50 | 5 | — | |
UXXQWNZSWRNFEM
|
6.8 | IC50 | 2 | — | |
RZOPCTSAJGVMBC
|
6.8 | IC50 | 2 | — | |
SAJFRQHNTSYGIH
|
6.8 | IC50 | 2 | — | |
RSDNMYGQEMFEDV
|
6.8 | IC50 | 2 | — | |
FNLMOWYVYCOJCX
|
6.8 | IC50 | 2 | — | |
MOQBQLRBTMTTNP
|
6.8 | IC50 | 2 | — | |
DUJLPWXXOJAVKA
|
6.7 | IC50 | 2 | — | |
RERINPGTUQBMDR
|
6.7 | IC50 | 2 | — | |
CEXHSRXBSHTSNU
|
6.7 | IC50 | 2 | — | |
FYEPWYBAIRUHTF
|
6.7 | IC50 | 2 | — | |
JBLHDYOCJVQGEP
|
6.7 | IC50 | 5 | — | |
OGLREAITVXTJOM
|
6.7 | IC50 | 2 | — | |
PVXYYWORFYROCX
|
6.7 | IC50 | 4 | — |