Target Details
| UniProt AC | Q03164 |
|---|---|
| Gene Symbol | KMT2A |
| Protein Name | Histone-lysine N-methyltransferase 2A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05965 (FYRC) PF05964 (FYRN) PF00628 (PHD) PF00856 (SET) PF02008 (zf-CXXC) PF13771 (zf-HC5HC2H) |
Summary
- Multi-target molecules 252
- Clinical molecules 0
- Avg pChEMBL 7.03
KEGG Pathways (4)
Associated Diseases (3)
Active Molecules (252)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YJMQZRJEJVTXJE
|
7.6 | IC50 | 2 | — | |
ZHYZCBJKPUJNCX
|
7.6 | IC50 | 2 | — | |
MEYYIZALDRYBJG
|
7.6 | Ki | 2 | — | |
WJGYXDBHCDMYQC
|
7.6 | IC50 | 2 | — | |
WYYACVUBSSTLHB
|
7.6 | IC50 | 2 | — | |
OSDQDWWAVUDZOY
|
7.6 | IC50 | 2 | — | |
QILXUBJKJXLPJR
|
7.6 | IC50 | 2 | — | |
BACRUGIGWRRCPL
|
7.6 | Kd | 2 | — | |
HWBBSTOZNJTCST
|
7.6 | IC50 | 5 | — | |
PRXLULUYVGAUHN
|
7.6 | IC50 | 2 | — | |
QFJNRXWVXGFRMJ
|
7.6 | IC50 | 2 | — | |
QFXSVAILBORUFA
|
7.6 | IC50 | 2 | — | |
SGSKCUULBFTJTH
|
7.6 | IC50 | 2 | — | |
VAXKDJXJCBGPOZ
|
7.5 | IC50 | 2 | — | |
WNZPPUDGOCDFHQ
|
7.5 | IC50 | 5 | — | |
IHHNJHMFVHNJBO
|
7.5 | IC50 | 2 | — | |
PSOJDGBGVBEYJX
|
7.5 | IC50 | 2 | — | |
GVUFUZRLWIDDCW
|
7.5 | IC50 | 2 | — | |
YITIAXSPNZIIEQ
|
7.5 | IC50 | 2 | — | |
JGYZPBXCLTVSLG
|
7.5 | IC50 | 2 | — | |
ZOQGZCVBPRNBEP
|
7.5 | IC50 | 2 | — | |
UUCBZFVZRYUNFK
|
7.4 | IC50 | 2 | — | |
KCTFIWDZXROTJT
|
7.4 | IC50 | 2 | — | |
QXVQPHOTRMOPJS
|
7.4 | IC50 | 2 | — | |
YRNWQOLFUAOQEK
|
7.4 | IC50 | 2 | — | |
NAQAQSQPMQDCCJ
|
7.4 | IC50 | 2 | — | |
PYVSJMIULSNDBE
|
7.4 | IC50 | 2 | — | |
QXVQPHOTRMOPJS
|
7.4 | IC50 | 2 | — | |
UPXZIGNTZNYNLJ
|
7.4 | IC50 | 2 | — | |
ZQYITMKVJCFUMK
|
7.4 | IC50 | 2 | — | |
BAGXALGFHCQJHH
|
7.4 | IC50 | 2 | — | |
KCTFIWDZXROTJT
|
7.4 | IC50 | 2 | — | |
CMLDSGMHBCTTQH
|
7.4 | IC50 | 2 | — | |
UETJRHPTKZEBKL
|
7.4 | IC50 | 2 | — | |
KCTFIWDZXROTJT
|
7.3 | IC50 | 2 | — | |
SFDROHXKTATJBI
|
7.3 | IC50 | 2 | — | |
BAOZMBPXQIZDNW
|
7.3 | IC50 | 2 | — | |
RSWJWQUYPRQBFS
|
7.3 | IC50 | 5 | — | |
ABZPYVVLYOUCEV
|
7.3 | IC50 | 2 | — | |
HDZDPXBIYCSDDH
|
7.3 | IC50 | 2 | — | |
LUFDPJMTRDADLV
|
7.3 | IC50 | 2 | — | |
RWMJXLQEZZOCBN
|
7.3 | IC50 | 2 | — | |
VJMSEJCFUWKXQR
|
7.3 | IC50 | 2 | — | |
BNFSVXBSRYHZTB
|
7.2 | IC50 | 5 | — | |
IOXMNCZSIBUWBK
|
7.2 | IC50 | 2 | — | |
AKMXHRWRBGESKY
|
7.2 | IC50 | 2 | — | |
BGABNIUBTFNMNB
|
7.2 | IC50 | 2 | — | |
KAVBMCHFVYVUGP
|
7.2 | IC50 | 2 | — | |
KJOQVBZBXKPYJX
|
7.2 | IC50 | 5 | — | |
ZCUAKOZUNBGFHR
|
7.2 | IC50 | 2 | — |