Target Details
| UniProt AC | Q03164 |
|---|---|
| Gene Symbol | KMT2A |
| Protein Name | Histone-lysine N-methyltransferase 2A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05965 (FYRC) PF05964 (FYRN) PF00628 (PHD) PF00856 (SET) PF02008 (zf-CXXC) PF13771 (zf-HC5HC2H) |
Summary
- Multi-target molecules 252
- Clinical molecules 0
- Avg pChEMBL 7.03
KEGG Pathways (4)
Associated Diseases (3)
Active Molecules (252)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MBFYNGBMAACLAT
|
9.3 | IC50 | 2 | — | |
XVEVAEBDYQDZRJ
|
9.3 | IC50 | 2 | — | |
ROBJDFLYWHJESD
|
9.1 | IC50 | 2 | — | |
QJWOBZCZCISQBL
|
9.0 | IC50 | 2 | — | |
AOGPBKJKSGZHDZ
|
8.6 | IC50 | 2 | — | |
BCIPILGGOSCOMC
|
8.5 | IC50 | 5 | — | |
PJMFCNODKBGQNV
|
8.5 | IC50 | 2 | — | |
HLVBKFBJGZIHHT
|
8.5 | Kd | 2 | — | |
DJHPKVNSQIOFKC
|
8.4 | IC50 | 2 | — | |
PTJOIPPVAWDZSV
|
8.3 | IC50 | 2 | — | |
RTZIJZSUBQDPEK
|
8.3 | IC50 | 2 | — | |
ANCOXZQAZPFGAR
|
8.3 | IC50 | 2 | — | |
SKALBDQRURDSRO
|
8.3 | IC50 | 2 | — | |
NTHBHLVHEBDGDP
|
8.2 | IC50 | 2 | — | |
ULYNNDWGUHSVCE
|
8.2 | IC50 | 2 | — | |
PKONCIPMLLIAIL
|
8.2 | IC50 | 2 | — | |
MACYWXUFQMTCBD
|
8.2 | IC50 | 2 | — | |
MWXGAMJNJKYTPA
|
8.2 | IC50 | 2 | — | |
PLYBGYMZTMVRST
|
8.2 | IC50 | 2 | — | |
SKALBDQRURDSRO
|
8.2 | IC50 | 2 | — | |
CQSKOHMINKNMTI
|
8.1 | IC50 | 2 | — | |
IOZUAULLLIHQBP
|
8.1 | IC50 | 2 | — | |
KMCCLTBDFVCDLQ
|
8.1 | IC50 | 2 | — | |
ZYADRCWVQPCKIY
|
8.1 | IC50 | 2 | — | |
LLVBFNANVRQGPY
|
8.1 | IC50 | 2 | — | |
BEHFFTBOQFMKCE
|
8.0 | IC50 | 2 | — | |
CKDLYAZOGRWEDP
|
8.0 | IC50 | 2 | — | |
VNGRFFKEZVSXII
|
8.0 | Kd | 2 | — | |
OZMZCHUIKIJUJP
|
8.0 | IC50 | 2 | — | |
UCJKXVRQFHYNKG
|
8.0 | IC50 | 2 | — | |
ZYADRCWVQPCKIY
|
7.9 | IC50 | 2 | — | |
LKCQRPVERQDLKW
|
7.9 | IC50 | 2 | — | |
NNIBWLKDWXOMEW
|
7.9 | IC50 | 5 | — | |
ZAIPJVQTYUSDTG
|
7.9 | IC50 | 5 | — | |
XNLFOGWQUFHWMA
|
7.9 | IC50 | 2 | — | |
VZVGYBWZKFBJTE
|
7.9 | IC50 | 2 | — | |
DETOMBLLEOZTMZ
|
7.8 | IC50 | 2 | — | |
MCSPTTKMVWDFHV
|
7.8 | IC50 | 2 | — | |
DZACSLYTXLZAAF
|
7.8 | IC50 | 2 | — | |
ZNCYDGWICNBNGY
|
7.8 | IC50 | 5 | — | |
KOHLMNSAZHTKAJ
|
7.8 | IC50 | 2 | — | |
VOEPLGKRDALOSS
|
7.8 | IC50 | 2 | — | |
YPEBLSPIUFKGDE
|
7.8 | IC50 | 2 | — | |
MQMLGCIPOBNMMG
|
7.8 | IC50 | 2 | — | |
PFDDMIFFNVKFIA
|
7.7 | IC50 | 2 | — | |
ZPVQIJIWGMKMQN
|
7.7 | IC50 | 2 | — | |
BAWZTNUTCPWRFJ
|
7.7 | IC50 | 5 | — | |
QOCGVCJRGIQEBR
|
7.7 | IC50 | 2 | — | |
ZIAHUDJHXDVKDL
|
7.7 | IC50 | 2 | — | |
HVYIAMBLIRZVRN
|
7.6 | IC50 | 2 | — |