Target Details
| UniProt AC | Q02880 |
|---|---|
| Gene Symbol | TOP2B |
| Protein Name | DNA topoisomerase 2-beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00204 (DNA_gyraseB) PF00521 (DNA_topoisoIV) PF08070 (DTHCT) PF02518 (HATPase_c) PF01751 (Toprim) PF16898 (TOPRIM_C) |
Summary
- Multi-target molecules 24
- Clinical molecules 0
- Avg pChEMBL 6.34
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (24)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LNMIYHCOSIHDEA
|
7.6 | IC50 | 3 | — | |
ASUGUQWIHMTFJL
|
6.8 | Kd | 18 | — | |
RADOMWSCHLMJFC
|
6.6 | IC50 | 2 | — | |
VJJPUSNTGOMMGY
|
6.6 | IC50 | 2 | — | |
XEKVSFQOGQZWKU
|
6.6 | IC50 | 2 | — | |
QULXAJAMUPGPBY
|
6.4 | IC50 | 2 | — | |
QULXAJAMUPGPBY
|
6.4 | IC50 | 2 | — | |
ZOGXKBMPGKLMPO
|
6.4 | IC50 | 2 | — | |
XEKVSFQOGQZWKU
|
6.3 | IC50 | 2 | — | |
DPZHKMWQVLEILB
|
6.3 | IC50 | 2 | — | |
ZJHZBDRZEZEDGB
|
6.3 | IC50 | 2 | — | |
OLNJLTFSGFZCKE
|
6.3 | IC50 | 2 | — | |
DXFOJQSWALTPJY
|
6.3 | IC50 | 2 | — | |
XEKVSFQOGQZWKU
|
6.3 | IC50 | 2 | — | |
QXXTYULODZEBMY
|
6.2 | IC50 | 2 | — | |
TXLRBFMVGQVAMM
|
6.1 | IC50 | 2 | — | |
MYSWGUAQZAJSOK
|
6.1 | IC50 | 6 | — | |
XSXKYRIANCDIFR
|
6.1 | IC50 | 2 | — | |
AGJYXSKRAATGBL
|
6.1 | IC50 | 2 | — | |
QULXAJAMUPGPBY
|
6.1 | IC50 | 2 | — | |
TXLRBFMVGQVAMM
|
6.1 | IC50 | 2 | — | |
IRTJFFVSCWKKTN
|
6.1 | IC50 | 2 | — | |
LMJFJIDLEAWOQJ
|
6.0 | Kd | 6 | — | |
LHFXYOYUZZPXSR
|
6.0 | IC50 | 2 | — |