Target Details
| UniProt AC | Q02779 |
|---|---|
| Gene Symbol | MAP3K10 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 10 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF14604 (SH3_9) |
Summary
- Multi-target molecules 33
- Clinical molecules 7
- Avg pChEMBL 7.04
KEGG Pathways (3)
Active Molecules (33)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OWRXHGAFWZFFCW
|
9.1 | Ki | 113 | — | |
HKSZLNNOFSGOKW
|
8.5 | Ki | 118 | — | |
NHHQJBCNYHBUSI
|
8.4 | Kd | 220 | — | |
UIARLYUEJFELEN
|
7.8 | Kd | 289 | Yes | |
MDAFGVXLBFQEJH
|
7.8 | IC50 | 4 | — | |
CVXZWDPKRAIHOI
|
7.7 | IC50 | 4 | — | |
UFLRHQRKTYVKGB
|
7.5 | IC50 | 4 | — | |
QKKIWEILHCXECO
|
7.4 | IC50 | 24 | — | |
KOZFSFOOLUUIGY
|
7.3 | IC50 | 26 | — | |
KOZFSFOOLUUIGY
|
7.3 | IC50 | 88 | Yes | |
OCMCHCVNRKLMAQ
|
7.3 | IC50 | 4 | — | |
APPXQUDJLJXULP
|
7.3 | IC50 | 47 | — | |
SCMLRESZJCKCTC
|
7.3 | IC50 | 7 | — | |
HKSZLNNOFSGOKW
|
7.3 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
7.3 | Kd | 213 | — | |
OUJZYQBEFNDJQN
|
7.1 | Ki | 71 | — | |
SIHPNVHZKXZMMW
|
7.0 | IC50 | 3 | — | |
JZTOUVBEZONDKA
|
6.9 | Ki | 80 | — | |
LRZYYIZFBXFSJB
|
6.9 | Ki | 69 | — | |
LYFDGRJCBMWOKJ
|
6.8 | IC50 | 3 | — | |
MZDKLVOWGIOKTN
|
6.7 | Ki | 80 | — | |
UYJNQQDJUOUFQJ
|
6.5 | Ki | 68 | — | |
NHDDTLMPCVOXFH
|
6.5 | IC50 | 16 | Yes | |
NBGYLHIDCLVBHE
|
6.4 | IC50 | 6 | Yes | |
GCIKSSRWRFVXBI
|
6.4 | Ki | 109 | Yes | |
SIXVRXARNAVBTC
|
6.3 | IC50 | 12 | — | |
CXQHYVUVSFXTMY
|
6.3 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.3 | Kd | 149 | — | |
CMAAJKFJPMUHEN
|
6.2 | IC50 | 3 | — | |
PRRYQINUAIQTFJ
|
6.2 | Ki | 11 | — | |
RHFIAUKMKYHHFA
|
6.1 | IC50 | 9 | — | |
BMGQWWVMWDBQGC
|
6.1 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.1 | Kd | 91 | Yes |