Target Details
| UniProt AC | Q02763 |
|---|---|
| Gene Symbol | TEK |
| Protein Name | Angiopoietin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF10430 (Ig_Tie2_1) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 507
- Clinical molecules 302
- Avg pChEMBL 7.5
KEGG Pathways (6)
Associated Diseases (3)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NWEIPABWNQPRCZ
|
7.2 | IC50 | 7 | Yes | |
YRSYWYSGZPRSOP
|
7.2 | IC50 | 2 | — | |
OSUPNTUMBGPMEA
|
7.2 | IC50 | 3 | — | |
ZPSQSBRNPLBDHP
|
7.2 | pIC50 | 3 | Yes | |
FMETVQKSDIOGPX
|
7.2 | pIC50 | 7 | Yes | |
STVKLDUINKMZFE
|
7.2 | pIC50 | 4 | Yes | |
XAIJULJJMLLWOQ
|
7.2 | IC50 | 2 | — | |
XZDKAVSSXNBWNJ
|
7.1 | pIC50 | 5 | Yes | |
ZIJIMHMKDXTURQ
|
7.1 | IC50 | 6 | Yes | |
OGKWTSFTGHKPIC
|
7.1 | IC50 | 3 | — | |
APPXQUDJLJXULP
|
7.1 | IC50 | 47 | — | |
FMIWNLDVSLITSM
|
7.1 | pIC50 | 2 | Yes | |
NOLVXPFFXLMLIM
|
7.1 | IC50 | 2 | — | |
SPMVMDHWKHCIDT
|
7.1 | IC50 | 30 | — | |
VZHPNWDSQYCLOK
|
7.1 | IC50 | 3 | — | |
RETUSTLIJKZUGV
|
7.1 | pIC50 | 5 | Yes | |
NMULSNNATHYGPZ
|
7.1 | IC50 | 3 | Yes | |
UFWXSGVSQZKZTR
|
7.1 | IC50 | 4 | — | |
UVNDVSUMHWZESZ
|
7.1 | pIC50 | 8 | Yes | |
QHQWGJPISLNJMT
|
7.1 | IC50 | 3 | Yes | |
NWUMNBBQSAYYPI
|
7.1 | IC50 | 2 | — | |
RGGYJEYZTPRESN
|
7.1 | IC50 | 6 | Yes | |
NJIPSDZQQSUQQF
|
7.0 | IC50 | 2 | — | |
KLEUWSFCKXAIKJ
|
7.0 | Kd | 2 | — | |
BIPPSOZOQMDQPZ
|
7.0 | IC50 | 4 | — | |
LHCIBQLPMCBTDW
|
7.0 | Kd | 3 | — | |
PNGAHMAIVIRYPV
|
7.0 | pIC50 | 3 | Yes | |
DYMJWJDJSBQQRF
|
7.0 | IC50 | 2 | — | |
STDSMFMGPYMGRQ
|
7.0 | pIC50 | 3 | Yes | |
ZXTNBCJQGUOHPF
|
7.0 | IC50 | 2 | — | |
SBLMCLDRWJNEJK
|
7.0 | IC50 | 17 | — | |
ZHGVDHRJPICWON
|
7.0 | pIC50 | 2 | Yes | |
FDVSOQRNTAPCHB
|
7.0 | pIC50 | 8 | Yes | |
FDVSOQRNTAPCHB
|
7.0 | pIC50 | 7 | Yes | |
GGMZFMQKFFREQV
|
7.0 | IC50 | 2 | — | |
UXYOQWHGYMKOQZ
|
7.0 | pIC50 | 2 | Yes | |
GWKIGGBPQCNPSU
|
7.0 | pIC50 | 3 | Yes | |
HRUYZDJOLIPWLW
|
7.0 | pIC50 | 5 | Yes | |
OKKAENUKIYEBBD
|
7.0 | pIC50 | 4 | Yes | |
UDCBEUBJXKUIRF
|
7.0 | pIC50 | 2 | Yes | |
UJBJAMOSBBJZBK
|
7.0 | IC50 | 6 | Yes | |
CUIYKFICQYRIMQ
|
6.9 | pIC50 | 3 | Yes | |
DXEWSKPRNSBDQR
|
6.9 | IC50 | 2 | — | |
FYIHXEFHXYJYLA
|
6.9 | pIC50 | 2 | Yes | |
KBJCTAIADOTYHC
|
6.9 | pIC50 | 8 | Yes | |
KKVYYGGCHJGEFJ
|
6.9 | IC50 | 6 | Yes | |
NQHMMDRPRXVCLT
|
6.9 | IC50 | 8 | Yes | |
PIQNNSKBFMKWGB
|
6.9 | pIC50 | 4 | Yes | |
QOKKLGWZLSTDCY
|
6.9 | pIC50 | 3 | Yes | |
PMZVFSAGPDDIJA
|
6.9 | IC50 | 3 | — |