Target Details
| UniProt AC | Q02763 |
|---|---|
| Gene Symbol | TEK |
| Protein Name | Angiopoietin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF10430 (Ig_Tie2_1) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 507
- Clinical molecules 302
- Avg pChEMBL 7.5
KEGG Pathways (6)
Associated Diseases (3)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UPGBUHOFLSJEEI
|
7.5 | pIC50 | 2 | Yes | |
JUPMOGJCVRJIHK
|
7.5 | pIC50 | 3 | Yes | |
KNXNQDZKPNJJEY
|
7.5 | pIC50 | 3 | Yes | |
YPTADYIVARXAPS
|
7.4 | pIC50 | 2 | Yes | |
SRNHAKVSFVSSPN
|
7.4 | IC50 | 8 | Yes | |
SXLHBXZCPKJTRT
|
7.4 | IC50 | 2 | — | |
BRXKGRHLVVRORC
|
7.4 | pIC50 | 2 | Yes | |
SSHDKAJDJAVHAF
|
7.4 | IC50 | 8 | Yes | |
OJRMOHAWDGZYFB
|
7.4 | IC50 | 2 | — | |
AQXIMVWUURMKKC
|
7.4 | pIC50 | 7 | Yes | |
AANHDPNKSQAGIM
|
7.4 | IC50 | 2 | — | |
KRICMVKKVCDVBV
|
7.4 | pIC50 | 7 | Yes | |
NYQWECLBSROSIH
|
7.4 | pIC50 | 3 | Yes | |
VHCQYUCVMXQFBY
|
7.4 | IC50 | 2 | — | |
AJCUOYPNGRYALV
|
7.4 | IC50 | 2 | — | |
BVMNEXLWCLAYGS
|
7.4 | pIC50 | 2 | Yes | |
CVMUHXWSBHMVGZ
|
7.4 | IC50 | 6 | Yes | |
GMVQPWCWWLPOQT
|
7.4 | IC50 | 3 | — | |
SVRMYHWEROXUTF
|
7.4 | pIC50 | 2 | Yes | |
VQRJYECHVOWPDV
|
7.4 | IC50 | 6 | Yes | |
JZSLVCXMHPNGNA
|
7.3 | IC50 | 5 | — | |
KMNCFOUKJYOZIF
|
7.3 | pIC50 | 7 | Yes | |
USFUHWQRVTVWKY
|
7.3 | IC50 | 2 | — | |
VHMGFCASMVCMMO
|
7.3 | pIC50 | 3 | Yes | |
CCUWZTRFTGLQCV
|
7.3 | IC50 | 5 | Yes | |
UHTHHESEBZOYNR
|
7.3 | pIC50 | 66 | Yes | |
LIMHWCZODBAXBC
|
7.3 | IC50 | 3 | — | |
FZQWDHPNNCNJFX
|
7.3 | IC50 | 2 | — | |
GPKUCJXJHXAHGN
|
7.3 | pIC50 | 3 | Yes | |
MXHHCGBNNWOCGV
|
7.3 | pIC50 | 3 | Yes | |
WGRSUBGGVRCDHQ
|
7.3 | pIC50 | 3 | Yes | |
KNKIKEKAVNITNK
|
7.3 | pIC50 | 3 | Yes | |
CZGMEOAMQWAJOY
|
7.3 | pIC50 | 15 | Yes | |
ISBXIYLTBRTLRK
|
7.3 | IC50 | 3 | — | |
RZDRBCYADHCOMG
|
7.2 | pIC50 | 3 | Yes | |
DVAKZOIIORDUJI
|
7.2 | pIC50 | 2 | Yes | |
UJWXPHLWGVGIBB
|
7.2 | IC50 | 4 | Yes | |
VTWWRKFUHCSCEW
|
7.2 | Kd | 19 | — | |
CQCCNBVEDUYZMC
|
7.2 | IC50 | 2 | — | |
PSDTVRBCPBZBIK
|
7.2 | pIC50 | 2 | Yes | |
DJCCECXADYTNDZ
|
7.2 | IC50 | 3 | — | |
RZYAXQPODGDVBT
|
7.2 | IC50 | 2 | — | |
ACOWAIUKUFGHLY
|
7.2 | pIC50 | 3 | Yes | |
OKAGZQCHRAGISN
|
7.2 | pIC50 | 2 | Yes | |
QSUZLYWASFSPHS
|
7.2 | pIC50 | 2 | Yes | |
HKSZLNNOFSGOKW
|
7.2 | IC50 | 408 | — | |
YOBIWCLAYQWPPW
|
7.2 | IC50 | 23 | — | |
ZPXXVJYFXNATQZ
|
7.2 | IC50 | 3 | — | |
FXQFQTDJCPCULX
|
7.2 | pIC50 | 3 | Yes | |
MZWALFBOTNMRTP
|
7.2 | IC50 | 7 | Yes |