Target Details
| UniProt AC | Q02763 |
|---|---|
| Gene Symbol | TEK |
| Protein Name | Angiopoietin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF10430 (Ig_Tie2_1) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 507
- Clinical molecules 302
- Avg pChEMBL 7.5
KEGG Pathways (6)
Associated Diseases (3)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DGRCFAYRKDYEMX
|
7.7 | IC50 | 7 | — | |
FXDWNCFVVOSWKM
|
7.7 | pIC50 | 5 | Yes | |
HKSZLNNOFSGOKW
|
7.7 | pIC50 | 49 | Yes | |
ODPGGGTTYSGTGO
|
7.7 | Kd | 153 | — | |
XLDWKHLQBFECEA
|
7.7 | pIC50 | 3 | Yes | |
ZDNWBLXKFNBSDR
|
7.7 | pIC50 | 3 | Yes | |
ANJMTRKKSQNBTH
|
7.7 | IC50 | 3 | — | |
KPFSWQACGQGZBB
|
7.7 | IC50 | 2 | — | |
MVCOAUNKQVWQHZ
|
7.7 | Kd | 54 | Yes | |
PAKQTWXBGSSCPQ
|
7.7 | IC50 | 2 | — | |
RRZDLEADQGXQKI
|
7.7 | IC50 | 2 | — | |
CBCKPZZVJQHROG
|
7.7 | IC50 | 5 | — | |
DADASRPKWOGKCU
|
7.7 | IC50 | 9 | — | |
NJRWVVJEQIMSFC
|
7.7 | IC50 | 2 | — | |
SWNPCLQLHUWVAZ
|
7.7 | pIC50 | 9 | Yes | |
HSAQBRJGYZIVJP
|
7.7 | pIC50 | 5 | Yes | |
ROJPTCGXRHNIRD
|
7.6 | IC50 | 2 | — | |
YJQJSZIDTDMDQM
|
7.6 | pIC50 | 2 | Yes | |
DEMGLABBZSLUOH
|
7.6 | IC50 | 3 | — | |
KJUCPVIVNLPLEE
|
7.6 | Kd | 10 | — | |
QLKGZBYGKCVLEX
|
7.6 | IC50 | 5 | Yes | |
TYNIZPFUWFETEF
|
7.6 | IC50 | 2 | — | |
GTDRUFDOKAMNII
|
7.6 | IC50 | 3 | — | |
JYLMIXWMBBGQSD
|
7.6 | IC50 | 3 | — | |
MKUGRPMZUYUAIX
|
7.6 | pIC50 | 3 | Yes | |
NJPIJBWGCOBYBH
|
7.6 | pIC50 | 3 | Yes | |
RKFUKWHBZZWJNX
|
7.6 | pIC50 | 4 | Yes | |
HTZHPXKKPOLGTR
|
7.6 | IC50 | 9 | — | |
ONSZEUCTVQJHOZ
|
7.6 | IC50 | 9 | — | |
UQHQUPSFNPQLNI
|
7.6 | pIC50 | 8 | Yes | |
LFYJXEXEFATBPN
|
7.6 | Kd | 2 | — | |
OZWMSXPIQVMFDE
|
7.6 | pIC50 | 8 | Yes | |
PXXIFHQHWGNCHG
|
7.6 | pIC50 | 2 | Yes | |
VIHXUAKPZPXVSW
|
7.6 | IC50 | 6 | Yes | |
XHHBBSIBRLADLF
|
7.6 | pIC50 | 3 | Yes | |
BTDHMLNFQMGPGD
|
7.5 | pIC50 | 3 | Yes | |
JGISZYJIPFCGCZ
|
7.5 | IC50 | 3 | — | |
KOXXIOJJABCMDV
|
7.5 | IC50 | 2 | — | |
ZEXJBANGHOAHDZ
|
7.5 | IC50 | 8 | Yes | |
ZYYNXHSAMWEIKK
|
7.5 | pIC50 | 4 | Yes | |
FCCZSKATTXDLOB
|
7.5 | pIC50 | 3 | Yes | |
HHKGVQGXRGQBBA
|
7.5 | IC50 | 4 | Yes | |
IZZAJZCFAZXNDC
|
7.5 | pIC50 | 6 | Yes | |
KERAXCVZALMMNG
|
7.5 | IC50 | 2 | — | |
PPELEVXKKDIBFP
|
7.5 | IC50 | 2 | — | |
KRCUBKFBOPSUJT
|
7.5 | pIC50 | 2 | Yes | |
XFYBEVQJFKVXIY
|
7.5 | IC50 | 2 | — | |
YTFRDKYCZHOSMM
|
7.5 | pIC50 | 4 | Yes | |
JLBAXNKYJZOYGQ
|
7.5 | pIC50 | 4 | Yes | |
LSYSLIJSKJGOJX
|
7.5 | pIC50 | 2 | Yes |