Target Details
| UniProt AC | Q02763 |
|---|---|
| Gene Symbol | TEK |
| Protein Name | Angiopoietin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF10430 (Ig_Tie2_1) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 507
- Clinical molecules 302
- Avg pChEMBL 7.5
KEGG Pathways (6)
Associated Diseases (3)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZTNZIYTUYLFXOO
|
8.0 | IC50 | 2 | — | |
BARYYLFEOIUPEY
|
7.9 | IC50 | 4 | Yes | |
FOOPCYOJMREECW
|
7.9 | IC50 | 5 | — | |
NWAUBAGBGOPJLF
|
7.9 | pIC50 | 51 | Yes | |
QQWUGDVOUVUTOY
|
7.9 | pIC50 | 231 | Yes | |
VSJXTUFWPAOYLC
|
7.9 | pIC50 | 11 | Yes | |
IGMQBINYIPIDJQ
|
7.9 | pIC50 | 9 | Yes | |
KIXJPVWFCZCXOL
|
7.9 | pIC50 | 4 | Yes | |
LGMDJFPPNVPECO
|
7.9 | pIC50 | 3 | Yes | |
UKSRSPVTFVLKRY
|
7.9 | pIC50 | 4 | Yes | |
AVHVXKAONMHRSS
|
7.9 | IC50 | 2 | — | |
BUBCSTHPMRUDOR
|
7.9 | IC50 | 2 | — | |
GHPCAIWYHJZRGR
|
7.9 | pIC50 | 3 | Yes | |
LKKLLNNNLUXMKW
|
7.9 | IC50 | 2 | — | |
UWBXUVYFALFCFH
|
7.9 | IC50 | 2 | — | |
NEJHRDWZMTYHKT
|
7.9 | IC50 | 3 | — | |
PATGADWTCHRVOQ
|
7.9 | pIC50 | 9 | Yes | |
KNDPXYAMINMLED
|
7.9 | IC50 | 11 | — | |
HVQYZYIFVKBRGI
|
7.9 | IC50 | 3 | — | |
VZRIBSCWFNIDIU
|
7.9 | IC50 | 3 | — | |
UVHLKFVTSZBBCD
|
7.8 | IC50 | 2 | — | |
XTPVNGSRCXLMPE
|
7.8 | IC50 | 3 | — | |
YNUAYENQUDYECY
|
7.8 | IC50 | 3 | — | |
ONIQOQHATWINJY
|
7.8 | IC50 | 25 | — | |
YNGDGIGDNVCQGR
|
7.8 | IC50 | 3 | — | |
FHDPQTHZTKXVCW
|
7.8 | pIC50 | 8 | Yes | |
GKOMRRDSXJXWIK
|
7.8 | pIC50 | 2 | Yes | |
NDXRDWNCKIAIEH
|
7.8 | IC50 | 3 | — | |
QFPRMYTURWHCEE
|
7.8 | pIC50 | 3 | Yes | |
TWOLOZGQZKJZKJ
|
7.8 | pIC50 | 7 | Yes | |
WLOVTHFKGZKSJV
|
7.8 | pIC50 | 2 | Yes | |
GHRNBCMJJKMYNR
|
7.8 | pIC50 | 4 | Yes | |
GOPWMXCRSJOJRB
|
7.8 | pIC50 | 2 | Yes | |
JDNWHCLQTRJTAJ
|
7.8 | IC50 | 6 | Yes | |
KCJAPLFLYYZXFD
|
7.8 | pIC50 | 2 | Yes | |
QPUJGBSZMTZOCB
|
7.8 | IC50 | 2 | — | |
UHEBDUAFKQHUBV
|
7.8 | pIC50 | 2 | Yes | |
VSMMGESTZLCGTL
|
7.8 | pIC50 | 2 | Yes | |
WXYYRQNZFXOQGI
|
7.8 | IC50 | 2 | — | |
DNZYFEKYHPAIRX
|
7.8 | IC50 | 3 | — | |
FICBCKOSWMLHMT
|
7.8 | IC50 | 3 | — | |
ZCGKVBJAWNXBSX
|
7.8 | IC50 | 3 | — | |
ZWVLMQTXUWMUII
|
7.8 | pIC50 | 9 | Yes | |
AOQSEIRRISHVNQ
|
7.8 | pIC50 | 3 | Yes | |
GXKSGTIXGWDSGJ
|
7.8 | IC50 | 12 | Yes | |
LGOFNTKAZMUZQC
|
7.8 | IC50 | 3 | — | |
LQCMQMYFSPQXKA
|
7.8 | pIC50 | 2 | Yes | |
NESXBRNDMQUVNG
|
7.8 | IC50 | 2 | — | |
AODUHZPEXFCKHF
|
7.7 | pIC50 | 2 | Yes | |
MTQVBIDLIJMPSF
|
7.7 | pIC50 | 2 | Yes |