Target Details
| UniProt AC | Q02763 |
|---|---|
| Gene Symbol | TEK |
| Protein Name | Angiopoietin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF10430 (Ig_Tie2_1) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 507
- Clinical molecules 302
- Avg pChEMBL 7.5
KEGG Pathways (6)
Associated Diseases (3)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GOEHHWWOYYPDII
|
8.3 | IC50 | 6 | Yes | |
PACMCHVNXJZGFE
|
8.3 | pIC50 | 2 | Yes | |
ODKIFGJQIHHLAP
|
8.3 | pIC50 | 2 | Yes | |
LILVTHVLIRBXAU
|
8.3 | pIC50 | 2 | Yes | |
NAHMZQCMCNMUAP
|
8.3 | pIC50 | 2 | Yes | |
MXEHLGSSZLWMBO
|
8.3 | IC50 | 3 | — | |
OTJLQOSBMKGOAA
|
8.3 | IC50 | 2 | — | |
IXIJKXSIADDKHR
|
8.2 | IC50 | 12 | — | |
UPABYWZSQBEEII
|
8.2 | IC50 | 6 | Yes | |
QFUIFWFJYBTUKA
|
8.2 | IC50 | 2 | — | |
SBRDWSXZGGLNQG
|
8.2 | IC50 | 2 | — | |
SLDNXLAQRVJNJO
|
8.2 | pIC50 | 5 | Yes | |
WVXNSAVVKYZVOE
|
8.2 | IC50 | 92 | — | |
YEVPZIUDTUZJGY
|
8.2 | pIC50 | 3 | Yes | |
SPSVDHUZUCNBNL
|
8.2 | IC50 | 2 | — | |
XOMNBLZPGBTSHU
|
8.2 | pIC50 | 2 | Yes | |
VCBGNDQGKNIBBK
|
8.2 | pIC50 | 6 | Yes | |
INFKEXSACBWFSL
|
8.2 | IC50 | 2 | — | |
VDQZIQXNPVFCAD
|
8.2 | pIC50 | 3 | Yes | |
KRAIQVKNMMQTGK
|
8.1 | pIC50 | 2 | Yes | |
QGMACHJORMNYMR
|
8.1 | pIC50 | 3 | Yes | |
OPPRLSONSGULSP
|
8.1 | pIC50 | 7 | Yes | |
CPTZKLNMWGFJMW
|
8.1 | IC50 | 3 | — | |
GNNDEPIMDAZHRQ
|
8.1 | IC50 | 6 | — | |
XDDKJJLWQBEZES
|
8.1 | pIC50 | 2 | Yes | |
AAAXBDFZRXKRPL
|
8.1 | IC50 | 6 | Yes | |
IAYJLHOAEWIYAY
|
8.1 | pIC50 | 4 | Yes | |
GYFAPMADUQCILZ
|
8.1 | IC50 | 5 | — | |
FKFACVZGGDYEHZ
|
8.1 | pIC50 | 5 | Yes | |
KEGATCOFPMKYRA
|
8.1 | pIC50 | 4 | Yes | |
QKPLUKMJEKRAJD
|
8.1 | pIC50 | 30 | Yes | |
ZUXFIRWLAQBCCS
|
8.1 | IC50 | 8 | Yes | |
GQWMMMAUWHLIBA
|
8.0 | IC50 | 2 | — | |
QDQFGRCUJGQRLD
|
8.0 | IC50 | 3 | — | |
UMGGFVAOWVEZEZ
|
8.0 | IC50 | 3 | — | |
AKAUSOQEQIKBNW
|
8.0 | IC50 | 2 | — | |
AQJFXYZAOCPIBG
|
8.0 | IC50 | 2 | — | |
BCZYLNWFHXDTAQ
|
8.0 | pIC50 | 3 | Yes | |
HHKWHHAJTWLRKG
|
8.0 | IC50 | 2 | — | |
KBJVFZCXZGSCFO
|
8.0 | IC50 | 3 | — | |
LIEYHNMAMBIXPW
|
8.0 | pIC50 | 3 | Yes | |
OHZQTNDZRUYHEH
|
8.0 | pIC50 | 3 | Yes | |
YHVHYWYQEFELOW
|
8.0 | IC50 | 44 | — | |
ZHARSIGHGZRJLM
|
8.0 | IC50 | 2 | — | |
LSVIBAPJYUUVJJ
|
8.0 | IC50 | 4 | — | |
LFDJFILTWUNEEP
|
8.0 | pIC50 | 6 | Yes | |
BOECRTNECUVVNV
|
8.0 | IC50 | 2 | — | |
CLLIAZGFVKRLRZ
|
8.0 | IC50 | 2 | — | |
HXHAJRMTJXHJJZ
|
8.0 | pIC50 | 52 | Yes | |
YJSFAHMGDRBZGH
|
8.0 | pIC50 | 16 | Yes |