Target Details
| UniProt AC | Q02763 |
|---|---|
| Gene Symbol | TEK |
| Protein Name | Angiopoietin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF10430 (Ig_Tie2_1) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 507
- Clinical molecules 302
- Avg pChEMBL 7.5
KEGG Pathways (6)
Associated Diseases (3)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OWBPDWHZXAEGMJ
|
8.7 | IC50 | 2 | — | |
SBSYQSASKXLENU
|
8.7 | IC50 | 5 | Yes | |
VOZWUTXGVBZOLP
|
8.7 | pIC50 | 2 | Yes | |
WBNNWMOEDXYOBE
|
8.7 | pIC50 | 2 | Yes | |
YEIASMOUYNOXGA
|
8.7 | IC50 | 5 | — | |
CLOKCIDZTVIDMJ
|
8.7 | pIC50 | 2 | Yes | |
DSRUNANRDDLTEB
|
8.7 | IC50 | 9 | — | |
SUXYGJZMCWKJJI
|
8.7 | IC50 | 26 | Yes | |
OPXHUNQHIWEERC
|
8.7 | IC50 | 2 | — | |
YZBMZVFTUOENSZ
|
8.6 | pIC50 | 2 | Yes | |
XLBQFFPUVVTFGK
|
8.6 | IC50 | 3 | — | |
PSQQJYVAJZSKPM
|
8.6 | IC50 | 2 | — | |
WYMDWWZXERLYKQ
|
8.6 | IC50 | 3 | — | |
IDBPJJQGJZOVMW
|
8.5 | pIC50 | 2 | Yes | |
ACZUPBJBDZROIE
|
8.5 | IC50 | 2 | — | |
CXDZGSNFZYGQSZ
|
8.5 | pIC50 | 4 | Yes | |
NFUYWPLTEOKUJO
|
8.5 | IC50 | 2 | — | |
UKICZFWMZQMZGK
|
8.5 | pIC50 | 3 | Yes | |
ZBJTXGNFKWUOFD
|
8.5 | IC50 | 2 | — | |
ZZOUIAPNOGIDSZ
|
8.5 | pIC50 | 2 | Yes | |
SEJGTFPOEJWEGG
|
8.5 | Kd | 149 | — | |
DZCUBLTYHLRLAF
|
8.5 | pIC50 | 2 | Yes | |
VWYXMUBOMREMIL
|
8.5 | IC50 | 2 | — | |
AEUDFMRQSRTMSH
|
8.5 | Kd | 4 | — | |
XXMJXRZJNGKMJK
|
8.5 | IC50 | 2 | — | |
DRWYYBMXZJLBHL
|
8.5 | IC50 | 3 | — | |
JPKSISIJPSXDLA
|
8.5 | pIC50 | 10 | Yes | |
KADQEUOYNAPXRD
|
8.5 | pIC50 | 3 | Yes | |
MPVGZUGXCQEXTM
|
8.5 | pIC50 | 61 | Yes | |
CEIFACIQCUXWSS
|
8.4 | IC50 | 2 | — | |
HTUPONJUVMCVCW
|
8.4 | IC50 | 6 | Yes | |
UVNBMNWTGOQKQF
|
8.4 | pIC50 | 8 | Yes | |
AIMHAFQTBGSBMF
|
8.4 | pIC50 | 3 | Yes | |
CRIVQNIFBMFYFY
|
8.4 | IC50 | 2 | — | |
FODDHYRWTNFLQO
|
8.4 | IC50 | 2 | — | |
IIHSBRSDVGUWER
|
8.4 | pIC50 | 2 | Yes | |
INFGJUQNPPGDNS
|
8.4 | IC50 | 2 | — | |
KGUBPBXMEHAZKB
|
8.4 | IC50 | 2 | — | |
LFLAFTJOXJJWMU
|
8.4 | pIC50 | 2 | Yes | |
NXSKYUVQJMCLKI
|
8.4 | IC50 | 2 | — | |
OKFRLDRBRRTBBF
|
8.4 | pIC50 | 2 | Yes | |
QTBWCSQGBMPECM
|
8.4 | pIC50 | 21 | Yes | |
TWTGVJCQGBDNIT
|
8.4 | pIC50 | 2 | Yes | |
WZPJVJBPNASYEY
|
8.4 | pIC50 | 2 | Yes | |
CASSAPBDIVDPCC
|
8.4 | pIC50 | 3 | Yes | |
VGXCATLWCWFSPS
|
8.4 | pIC50 | 3 | Yes | |
LSWBBDJKWCZRAP
|
8.3 | pIC50 | 2 | Yes | |
OOZBLQPABHWRKB
|
8.3 | IC50 | 3 | — | |
DCFCBTICZZTNCX
|
8.3 | pIC50 | 2 | Yes | |
GMVQPWCWWLPOQT
|
8.3 | IC50 | 9 | Yes |