Target Details
| UniProt AC | Q02763 |
|---|---|
| Gene Symbol | TEK |
| Protein Name | Angiopoietin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF10430 (Ig_Tie2_1) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 507
- Clinical molecules 302
- Avg pChEMBL 7.5
KEGG Pathways (6)
Associated Diseases (3)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VMZBKTOJOWBBSN
|
6.3 | IC50 | 2 | — | |
WCRYRBRNFCXTTR
|
6.3 | pIC50 | 4 | Yes | |
DWCZEZXJZXJTHE
|
6.3 | pIC50 | 6 | Yes | |
SPDICIKFASBCHA
|
6.3 | pIC50 | 2 | Yes | |
VOPNWXZDJKCCRE
|
6.3 | pIC50 | 7 | Yes | |
ZGTHJDQZGGIPLL
|
6.3 | IC50 | 5 | Yes | |
AECDBHGVIIRMOI
|
6.3 | IC50 | 7 | — | |
KKUNUMXHGLIOMX
|
6.3 | IC50 | 3 | — | |
ZQXWSHOYNMQRDD
|
6.3 | pIC50 | 4 | Yes | |
DJCDHWXQLRMRTB
|
6.2 | IC50 | 5 | — | |
FFNIWOOLZGAOAB
|
6.2 | pIC50 | 8 | Yes | |
FRQGIFZNGIECRT
|
6.2 | IC50 | 2 | — | |
KRYULLMPWHIEHI
|
6.2 | IC50 | 2 | — | |
PHWICBBDBJYOQR
|
6.2 | pIC50 | 3 | Yes | |
HJVFTUSVRMGBLM
|
6.2 | IC50 | 7 | — | |
VRWFLNVDDMVVDA
|
6.2 | IC50 | 7 | — | |
MYSJNRWPLKEUQT
|
6.2 | pIC50 | 3 | Yes | |
SKNUELOYQKBUOU
|
6.2 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
6.2 | Kd | 289 | Yes | |
CYXVEZJWVJIFPJ
|
6.2 | pIC50 | 4 | Yes | |
DAZCBQNFGSWSQG
|
6.2 | pIC50 | 8 | Yes | |
LYADGAGFYYXXIO
|
6.2 | IC50 | 82 | — | |
DIOOREPVPOCQKL
|
6.2 | pIC50 | 4 | Yes | |
HJWSKMQXMBSGEX
|
6.2 | IC50 | 2 | — | |
IFTCXKUSJMWVRD
|
6.2 | pIC50 | 7 | Yes | |
WPGZZMRHHXVHEX
|
6.2 | pIC50 | 2 | Yes | |
YISMQBFJYDFMAL
|
6.1 | IC50 | 46 | — | |
CJAOTOWETHYRND
|
6.1 | IC50 | 5 | — | |
OJFKUJDRGJSAQB
|
6.1 | IC50 | 17 | — | |
RKGNVOKYSGKVQZ
|
6.1 | pIC50 | 7 | Yes | |
DPYASQWYHILTBI
|
6.1 | pIC50 | 6 | Yes | |
KSBCGWKXTJXPLL
|
6.1 | IC50 | 3 | — | |
XEGSWNKCRGYRFG
|
6.1 | IC50 | 3 | — | |
BSBQPLUISHJULY
|
6.1 | IC50 | 11 | — | |
ILOAUSWXRCKWFH
|
6.1 | IC50 | 3 | Yes | |
GEPKFPGFWUHVLZ
|
6.1 | pIC50 | 6 | Yes | |
PIOFIWWMFVHCRR
|
6.0 | IC50 | 2 | — | |
CXUVPVMNMZKERT
|
6.0 | pIC50 | 3 | Yes | |
AOUMXCXOJGAKLX
|
6.0 | pIC50 | 3 | Yes | |
KDKUVYLMPJIGKA
|
6.0 | Kd | 91 | Yes | |
QBRQTJMZEYORSP
|
6.0 | Kd | 12 | — | |
GLBZSOQDAOLMGC
|
6.0 | IC50 | 23 | Yes | |
HHZIURLSWUIHRB
|
6.0 | Kd | 57 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
SYZJSPFCXVXDAA
|
6.0 | IC50 | 2 | — | |
BMGGDZTXJBWQCN
|
Clinical | TTD_MultiTarget | 2 | Yes | |
CAQLNQYCCKYWJX
|
Clinical | TTD_MultiTarget | 5 | Yes | |
CXJQAZDGOBZGLJ
|
Clinical | TTD_MultiTarget | 4 | Yes | |
CZUVMGAHFHQKLM
|
Clinical | TTD_MultiTarget | 3 | Yes | |
FLGQTDLHJSQLIG
|
Clinical | TTD_MultiTarget | 2 | Yes |