Target Details
| UniProt AC | Q02763 |
|---|---|
| Gene Symbol | TEK |
| Protein Name | Angiopoietin-1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF10430 (Ig_Tie2_1) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 507
- Clinical molecules 302
- Avg pChEMBL 7.5
KEGG Pathways (6)
Associated Diseases (3)
Active Molecules (507)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YULUVWHIOGBTPX
|
9.7 | pIC50 | 4 | Yes | |
NUWGRQLPQIXMCW
|
9.6 | IC50 | 2 | — | |
DTIBDUZHSDASKY
|
9.6 | IC50 | 2 | — | |
XMICLSPUPFMDHT
|
9.5 | IC50 | 2 | — | |
WYLBYVHRCHPXRQ
|
9.4 | IC50 | 3 | — | |
JRGLHUFNZUQJNB
|
9.3 | IC50 | 2 | — | |
VCDOUBNPUAACRA
|
9.3 | pIC50 | 2 | Yes | |
CEIYRBYXRSULDG
|
9.3 | pIC50 | 4 | Yes | |
RNHWXYKRVZUXGO
|
9.3 | pIC50 | 4 | Yes | |
WUBFAXNVDMCVIO
|
9.3 | pIC50 | 12 | Yes | |
PKFMTQRFZPFQOL
|
9.2 | pIC50 | 4 | Yes | |
YBUFHSXYBABPHF
|
9.2 | IC50 | 3 | — | |
MPASHPJAIUOWCK
|
9.2 | IC50 | 9 | — | |
UBPYILGKFZZVDX
|
9.2 | pIC50 | 130 | Yes | |
MIIRGIJHJBFFEA
|
9.1 | IC50 | 3 | — | |
IEIGLLZCPLOVEA
|
9.1 | IC50 | 2 | — | |
SQQPRORGDVPLSI
|
9.1 | IC50 | 4 | — | |
MLDQJTXFUGDVEO
|
9.1 | IC50 | 85 | Yes | |
BIGLUOGTKFYENL
|
9.0 | pIC50 | 2 | Yes | |
CKFIBJSVBPYSCR
|
9.0 | IC50 | 2 | — | |
CPZZPVRAQQJBTN
|
9.0 | pIC50 | 2 | Yes | |
CREAAGUFOMLCKF
|
9.0 | pIC50 | 3 | Yes | |
DJNWXYTWORPJNI
|
9.0 | pIC50 | 4 | Yes | |
FDWJEDYUZLTROC
|
9.0 | pIC50 | 2 | Yes | |
GGIPEVUWPMVPNG
|
9.0 | IC50 | 5 | Yes | |
LXBUSRPKZONHPE
|
9.0 | pIC50 | 4 | Yes | |
MQRYORPEARKGSY
|
9.0 | pIC50 | 4 | Yes | |
NKKSIIYIDSJFSX
|
9.0 | pIC50 | 3 | Yes | |
OHHGYJBFPVJURR
|
9.0 | IC50 | 2 | — | |
OQKMFDJSKWESCR
|
9.0 | IC50 | 4 | Yes | |
QSIAXFKUFXOHHK
|
9.0 | IC50 | 5 | Yes | |
XBINIPRQWSOQIE
|
9.0 | pIC50 | 4 | Yes | |
ZVIWALRWYYSHSU
|
9.0 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
9.0 | IC50 | 154 | — | |
MZWXPLVBKPHKNC
|
9.0 | pIC50 | 2 | Yes | |
FLYHDJWABMRYPV
|
8.9 | IC50 | 2 | — | |
BYYYCNUDMZSOGS
|
8.9 | pIC50 | 5 | Yes | |
DQHFKDYMNMRFQA
|
8.9 | pIC50 | 2 | Yes | |
YHYJQEMFCWJMSJ
|
8.9 | pIC50 | 2 | Yes | |
UTVABCSMEKUFLJ
|
8.9 | pIC50 | 7 | Yes | |
DZSUJUOJJJCWGG
|
8.8 | pIC50 | 55 | Yes | |
FNHKPVJBJVTLMP
|
8.8 | IC50 | 29 | — | |
WYSIIHBXZUVHPY
|
8.8 | pIC50 | 2 | Yes | |
PBYFXEFTMBEMLE
|
8.8 | IC50 | 2 | — | |
FCPPQNZGDIZFLT
|
8.7 | pIC50 | 3 | Yes | |
FGZIONRFHVNRJB
|
8.7 | IC50 | 3 | — | |
FOEQINTXCQEBGE
|
8.7 | IC50 | 2 | — | |
JXKDTYDBDDKIPY
|
8.7 | IC50 | 5 | Yes | |
MQCFWAKOIXTUQK
|
8.7 | pIC50 | 2 | Yes | |
NPUAKRMYWJOTLS
|
8.7 | IC50 | 2 | — |