Target Details
| UniProt AC | Q02156 |
|---|---|
| Gene Symbol | PRKCE |
| Protein Name | Protein kinase C epsilon type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 423
- Clinical molecules 146
- Avg pChEMBL 7.28
KEGG Pathways (13)
- AGE-RAGE signaling pathway in diabetic complications
- Aldosterone synthesis and secretion
- Apelin signaling pathway
- Fc gamma R-mediated phagocytosis
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- MicroRNAs in cancer
- Shigellosis
- Sphingolipid signaling pathway
- Tight junction
- Type II diabetes mellitus
- Vascular smooth muscle contraction
- cGMP-PKG signaling pathway
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HIUHVDROHDSKTC
|
6.2 | Ki | 20 | — | |
ORNADCNXUPZOQN
|
6.2 | IC50 | 15 | — | |
AXTAPYRUEKNRBA
|
6.1 | IC50 | 24 | — | |
FVNQTIFQMVXLGJ
|
6.1 | Ki | 3 | — | |
VSSNHBWGDBKVPE
|
6.1 | IC50 | 2 | — | |
WSXYBDKZFNJOTP
|
6.1 | IC50 | 12 | Yes | |
MRBNLCLXWRXFJX
|
6.1 | IC50 | 15 | — | |
WUXPTIWFTBYPCX
|
6.1 | Ki | 5 | Yes | |
CMPYJCKDXNDOGF
|
6.1 | IC50 | 2 | — | |
GHRBXKFGXPOEGA
|
6.0 | IC50 | 12 | Yes | |
VYXIZKJRRNWQAK
|
6.0 | IC50 | 6 | — | |
LADIDEKFWKOIAL
|
6.0 | IC50 | 2 | — | |
SSMSJTVEHMWTFZ
|
6.0 | IC50 | 6 | — | |
SSMSJTVEHMWTFZ
|
6.0 | IC50 | 6 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
LWSORTKUYSYDMP
|
6.0 | IC50 | 12 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NKANXQFJJICGDU
|
6.0 | IC50 | 35 | Yes | |
RELJBNLDXPSLLS
|
6.0 | IC50 | 6 | — | |
UUCJUCRTIKZRFG
|
6.0 | IC50 | 12 | Yes | |
XBFAFSAUQFDEOK
|
6.0 | IC50 | 5 | — | |
XYUFCXJZFZPEJD
|
6.0 | IC50 | 5 | — |