Target Details
| UniProt AC | Q02156 |
|---|---|
| Gene Symbol | PRKCE |
| Protein Name | Protein kinase C epsilon type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 423
- Clinical molecules 146
- Avg pChEMBL 7.28
KEGG Pathways (13)
- AGE-RAGE signaling pathway in diabetic complications
- Aldosterone synthesis and secretion
- Apelin signaling pathway
- Fc gamma R-mediated phagocytosis
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- MicroRNAs in cancer
- Shigellosis
- Sphingolipid signaling pathway
- Tight junction
- Type II diabetes mellitus
- Vascular smooth muscle contraction
- cGMP-PKG signaling pathway
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KQUBTSBQLPIFSM
|
6.4 | IC50 | 5 | — | |
MQFYZWYYZGTHAN
|
6.4 | IC50 | 14 | — | |
ARKNUCQRPYIUMU
|
6.4 | IC50 | 6 | — | |
GDZULWKNFKCRJP
|
6.4 | IC50 | 7 | — | |
HHLKZSJXDAZIGG
|
6.4 | IC50 | 10 | Yes | |
JQGRMZUVGWRDIV
|
6.4 | IC50 | 6 | — | |
SNQKPKFVSANKFP
|
6.4 | IC50 | 6 | — | |
FSPDDRAYNYPNIF
|
6.4 | IC50 | 2 | — | |
FSPDDRAYNYPNIF
|
6.4 | IC50 | 2 | — | |
IYKCWOIZNVHUMI
|
6.4 | Ki | 5 | Yes | |
NFRKACJUZYOBMM
|
6.4 | Ki | 5 | Yes | |
UNULBQHMZBESJQ
|
6.4 | IC50 | 4 | — | |
KAJXOWFGKYKMMZ
|
6.4 | IC50 | 26 | Yes | |
ZFNQOYBHHLGQDV
|
6.3 | IC50 | 12 | Yes | |
PQWWKDOKHDWZBH
|
6.3 | IC50 | 6 | — | |
PQWWKDOKHDWZBH
|
6.3 | IC50 | 6 | — | |
BMBIKZHGTPMMMM
|
6.3 | IC50 | 14 | — | |
KLYPYTHLYUUKMT
|
6.3 | Ki | 4 | — | |
CPRVBHBRBVVLHL
|
6.3 | IC50 | 11 | — | |
SWZFTDYOTKYQHS
|
6.3 | IC50 | 2 | — | |
RSTWARDIGORXQU
|
6.3 | Ki | 5 | Yes | |
ATBAETXFFCOZOY
|
6.3 | IC50 | 39 | — | |
CCRCRSXDKXZDGK
|
6.3 | IC50 | 12 | Yes | |
WOFBHAKTZOZODW
|
6.3 | IC50 | 6 | — | |
IDVIOLNZWSXZGL
|
6.3 | Ki | 5 | Yes | |
PXONMVAMARNSJO
|
6.3 | Ki | 4 | — | |
DRTOCQUQJDNMBT
|
6.3 | IC50 | 3 | — | |
HFNKQEVNSGCOJV
|
6.3 | Kd | 65 | — | |
JSPAUBUYPPZXSG
|
6.3 | Ki | 17 | Yes | |
NTRDTMDMDUVYSM
|
6.3 | IC50 | 3 | — | |
ORNADCNXUPZOQN
|
6.3 | IC50 | 15 | — | |
BMGQWWVMWDBQGC
|
6.3 | Kd | 147 | Yes | |
OYPYXQXNEBSSGB
|
6.3 | Ki | 8 | Yes | |
NEGCBIBMPAHBIM
|
6.3 | IC50 | 12 | Yes | |
BAQFZMFDZMQJAM
|
6.2 | IC50 | 12 | Yes | |
RFUHKEPWGZUNBG
|
6.2 | IC50 | 4 | — | |
LASNFRKYDHLWNQ
|
6.2 | IC50 | 3 | — | |
TXBFOGDMTCNBBT
|
6.2 | IC50 | 12 | Yes | |
QQKKPWJFHBFCTH
|
6.2 | IC50 | 10 | Yes | |
TWUWFRLZDWDJLT
|
6.2 | Ki | 10 | Yes | |
ZCBUQCWBWNUWSU
|
6.2 | IC50 | 59 | — | |
ZUKHVOLIPVGCHQ
|
6.2 | Ki | 10 | Yes | |
JHWNRWTWKSNTOD
|
6.2 | IC50 | 4 | — | |
HLXIFVDYTGEUJV
|
6.2 | IC50 | 15 | Yes | |
KPJDEGAKXAUVAC
|
6.2 | Ki | 15 | Yes | |
QHZHJSWWHXUNNZ
|
6.2 | IC50 | 2 | — | |
MGLBGUZLARZAOR
|
6.2 | IC50 | 4 | — | |
QRBLWZIADYBYNA
|
6.2 | IC50 | 5 | — | |
WLEQZZURIGPVJT
|
6.2 | Ki | 3 | — | |
CWFIQHQECWPWQG
|
6.2 | IC50 | 16 | Yes |