Target Details
| UniProt AC | Q02156 |
|---|---|
| Gene Symbol | PRKCE |
| Protein Name | Protein kinase C epsilon type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 423
- Clinical molecules 146
- Avg pChEMBL 7.28
KEGG Pathways (13)
- AGE-RAGE signaling pathway in diabetic complications
- Aldosterone synthesis and secretion
- Apelin signaling pathway
- Fc gamma R-mediated phagocytosis
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- MicroRNAs in cancer
- Shigellosis
- Sphingolipid signaling pathway
- Tight junction
- Type II diabetes mellitus
- Vascular smooth muscle contraction
- cGMP-PKG signaling pathway
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OXEOHAXVZADDOC
|
6.6 | IC50 | 12 | Yes | |
PXONMVAMARNSJO
|
6.6 | Ki | 4 | — | |
YSVVBGPTTSJYPA
|
6.6 | IC50 | 12 | Yes | |
NIUBYBAPAVVDMG
|
6.6 | IC50 | 6 | — | |
NIUBYBAPAVVDMG
|
6.6 | IC50 | 6 | — | |
QXQGSOMQKZFIRY
|
6.6 | IC50 | 10 | — | |
WOFBHAKTZOZODW
|
6.6 | IC50 | 6 | — | |
BNAXHIOTDMDOLF
|
6.6 | IC50 | 6 | — | |
JISUVVYQUNDVBH
|
6.6 | IC50 | 4 | — | |
KLTAXINXABHYMC
|
6.6 | IC50 | 5 | — | |
KOZFSFOOLUUIGY
|
6.6 | IC50 | 26 | — | |
SSZFVGXDYBMVDD
|
6.6 | IC50 | 12 | Yes | |
JOOTZGPUMCZHLH
|
6.6 | IC50 | 5 | — | |
PBCZSGKMGDDXIJ
|
6.6 | IC50 | 12 | Yes | |
CKJRKRPDNLRZPQ
|
6.6 | IC50 | 6 | — | |
LAOIBIIMKUINJL
|
6.6 | IC50 | 12 | Yes | |
ZYVVHWBUHYZJFE
|
6.6 | Ki | 3 | Yes | |
CKJRKRPDNLRZPQ
|
6.6 | IC50 | 7 | — | |
IXOVKVHWGKDXKQ
|
6.6 | IC50 | 12 | Yes | |
BRZYOTMFHLERHD
|
6.5 | Ki | 17 | Yes | |
JOOTZGPUMCZHLH
|
6.5 | IC50 | 5 | — | |
MDRQBBNTQCZOBR
|
6.5 | IC50 | 6 | — | |
MDRQBBNTQCZOBR
|
6.5 | IC50 | 6 | — | |
TXVBBLNFLUZGIT
|
6.5 | IC50 | 6 | — | |
XRZURBBBXNHUNO
|
6.5 | IC50 | 7 | Yes | |
GNIYOZALILMSSH
|
6.5 | Ki | 3 | — | |
KTTKZYWEKGBVIX
|
6.5 | IC50 | 3 | — | |
KTTKZYWEKGBVIX
|
6.5 | IC50 | 3 | — | |
RRGGCASWPGLJTK
|
6.5 | Ki | 3 | — | |
UIOPZRFPFXYNME
|
6.5 | Ki | 3 | — | |
XNKIVXYFRPYKHO
|
6.5 | IC50 | 12 | Yes | |
YRTMRGPNXUUDTD
|
6.5 | IC50 | 5 | — | |
FNTXTLNLTQPVBJ
|
6.5 | IC50 | 6 | — | |
NNVINYYJNCKGRA
|
6.5 | IC50 | 5 | — | |
PQWWKDOKHDWZBH
|
6.5 | IC50 | 6 | — | |
TVIALAOHRQNPOI
|
6.5 | IC50 | 12 | Yes | |
KCXYCCAYSVRIQM
|
6.5 | Ki | 2 | — | |
VNPLXDZLURAZHZ
|
6.5 | IC50 | 5 | — | |
IYOZTVGMEWJPKR
|
6.5 | IC50 | 5 | — | |
ZOGSVRRXRLSQNC
|
6.5 | IC50 | 6 | — | |
HPCPUHOULFPBCQ
|
6.5 | IC50 | 12 | Yes | |
JDZXLEPJWLCESI
|
6.5 | IC50 | 12 | Yes | |
PHOVPHVCAJYUNY
|
6.5 | IC50 | 3 | — | |
RHBWAFDCVFMIFK
|
6.5 | IC50 | 12 | Yes | |
RPLXVENRWORMRX
|
6.4 | IC50 | 12 | Yes | |
OVJZHEDXGAPGDA
|
6.4 | IC50 | 3 | — | |
OVJZHEDXGAPGDA
|
6.4 | IC50 | 5 | — | |
BIIVYFLTOXDAOV
|
6.4 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
6.4 | Kd | 82 | Yes | |
HTALWVZQUMMIDH
|
6.4 | Ki | 3 | — |