Target Details
| UniProt AC | Q02156 |
|---|---|
| Gene Symbol | PRKCE |
| Protein Name | Protein kinase C epsilon type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 423
- Clinical molecules 146
- Avg pChEMBL 7.28
KEGG Pathways (13)
- AGE-RAGE signaling pathway in diabetic complications
- Aldosterone synthesis and secretion
- Apelin signaling pathway
- Fc gamma R-mediated phagocytosis
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- MicroRNAs in cancer
- Shigellosis
- Sphingolipid signaling pathway
- Tight junction
- Type II diabetes mellitus
- Vascular smooth muscle contraction
- cGMP-PKG signaling pathway
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BJNQKVADRDIKFO
|
7.3 | Ki | 6 | Yes | |
JSXUDEUMWQFINT
|
7.3 | Ki | 3 | — | |
ZDFZJOAXAPUMLZ
|
7.2 | IC50 | 3 | — | |
QMYFYCSCELQGHP
|
7.2 | IC50 | 7 | Yes | |
WMOCKUYLGCVFJM
|
7.2 | Ki | 3 | — | |
XHUGZQWFSKJGAZ
|
7.2 | Ki | 3 | — | |
DVMQYKHCZLPSAP
|
7.2 | IC50 | 5 | — | |
XXIWRTOLXWAEJC
|
7.2 | IC50 | 13 | Yes | |
TUBBFDZWFNUZLH
|
7.2 | IC50 | 12 | Yes | |
NRUVICOXXLOXCB
|
7.2 | IC50 | 13 | Yes | |
MGMNDPRNDCWSMZ
|
7.2 | IC50 | 12 | Yes | |
HFPUIOYUZROFHG
|
7.1 | IC50 | 6 | — | |
HOWICUYRWBCICG
|
7.1 | IC50 | 6 | — | |
PKUWFMAWUYFHHA
|
7.1 | Ki | 3 | — | |
UWFSHWFUBYEFAT
|
7.1 | IC50 | 6 | — | |
GRENHRYHWHSBLM
|
7.1 | IC50 | 12 | Yes | |
KDIRIFZBLUSLJU
|
7.1 | Ki | 5 | — | |
SFDFKLDQKSPRHB
|
7.1 | IC50 | 15 | Yes | |
CYRPAUWSHGGREB
|
7.1 | Ki | 8 | Yes | |
GIVLJYSTNKNCGZ
|
7.1 | IC50 | 4 | — | |
LGCKGDRUTNACTA
|
7.1 | IC50 | 11 | — | |
NMSQMKXWQOPPRS
|
7.1 | Ki | 3 | — | |
OFPFIAWWDTYSBZ
|
7.1 | Ki | 15 | Yes | |
RHLRPKGACJKWPF
|
7.1 | IC50 | 12 | Yes | |
STEGBXHZVWLLAP
|
7.1 | IC50 | 6 | — | |
UXKZMYMPEYJJKA
|
7.1 | IC50 | 5 | — | |
GEATXDJAPAHPTP
|
7.1 | IC50 | 10 | — | |
GGQAEINRBKFRGZ
|
7.1 | IC50 | 15 | Yes | |
ZZKAMKCYEYGTEB
|
7.1 | IC50 | 4 | — | |
MVQGUYKZTHVOEH
|
7.1 | Ki | 8 | Yes | |
NHDDTLMPCVOXFH
|
7.1 | IC50 | 16 | Yes | |
OMTMFLTXXIJRAC
|
7.0 | Ki | 3 | — | |
SXDPQGRNHSLZPC
|
7.0 | IC50 | 18 | — | |
MQCCJEYZKWZQHU
|
7.0 | IC50 | 15 | Yes | |
YSVVBGPTTSJYPA
|
7.0 | IC50 | 13 | Yes | |
DPQYCBYVJBHECV
|
7.0 | Ki | 3 | — | |
OWJIKBAZUBPKGN
|
7.0 | IC50 | 6 | — | |
OWJIKBAZUBPKGN
|
7.0 | IC50 | 7 | — | |
PFAZIMNYEBJHOA
|
7.0 | IC50 | 12 | Yes | |
XRFOMFNAMTYCFF
|
7.0 | IC50 | 12 | Yes | |
YUAWUNMKPARPJD
|
7.0 | IC50 | 14 | Yes | |
INDMCILJGPHHCG
|
7.0 | Ki | 3 | — | |
AXRCEOKUDYDWLF
|
7.0 | IC50 | 31 | — | |
FOPORVBLOTVXEK
|
7.0 | Ki | 5 | — | |
LPIHDMXDUPXXEU
|
7.0 | IC50 | 6 | — | |
LRHWSAFUUBKSML
|
7.0 | Ki | 5 | — | |
KOZFSFOOLUUIGY
|
6.9 | IC50 | 15 | Yes | |
DAGKXAWMGQZKFD
|
6.9 | IC50 | 4 | — | |
DLMIREIQJNSNMF
|
6.9 | Ki | 3 | — | |
OBNHABKOCPUFDD
|
6.9 | Ki | 3 | — |