Target Details
| UniProt AC | Q02156 |
|---|---|
| Gene Symbol | PRKCE |
| Protein Name | Protein kinase C epsilon type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 423
- Clinical molecules 146
- Avg pChEMBL 7.28
KEGG Pathways (13)
- AGE-RAGE signaling pathway in diabetic complications
- Aldosterone synthesis and secretion
- Apelin signaling pathway
- Fc gamma R-mediated phagocytosis
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- MicroRNAs in cancer
- Shigellosis
- Sphingolipid signaling pathway
- Tight junction
- Type II diabetes mellitus
- Vascular smooth muscle contraction
- cGMP-PKG signaling pathway
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GQCWIZZVARXZGR
|
7.5 | IC50 | 6 | — | |
GQCWIZZVARXZGR
|
7.5 | IC50 | 6 | — | |
SMOYJWUKHYTHIN
|
7.5 | Ki | 2 | — | |
XXDWSQPJTJZKSJ
|
7.5 | IC50 | 12 | Yes | |
ZMHXVAQNZDUNOG
|
7.5 | IC50 | 6 | — | |
ZZSBPGIGIUFJRA
|
7.5 | IC50 | 15 | Yes | |
FELQRVDTGNDOSI
|
7.5 | IC50 | 15 | Yes | |
SIWILCBNYOGJQH
|
7.5 | Ki | 4 | — | |
IPBIYLHQBHMHCN
|
7.5 | Ki | 2 | — | |
MYOUXQLHWTWXON
|
7.5 | IC50 | 16 | Yes | |
UHIFMIXIMAHXIB
|
7.5 | IC50 | 6 | — | |
YDZJEODKNRAYMA
|
7.5 | IC50 | 12 | Yes | |
COPQMLDDHGHTAG
|
7.5 | Ki | 2 | — | |
FWEDWNSLCBHVQT
|
7.5 | IC50 | 5 | — | |
HSZCSAUAGLABDS
|
7.5 | Ki | 5 | — | |
PKUWFMAWUYFHHA
|
7.5 | Ki | 3 | — | |
XUTMONHBGYHWES
|
7.5 | Ki | 5 | — | |
ZYUGNHPOVKADFZ
|
7.5 | IC50 | 11 | — | |
HPBJQOWLAKYNDM
|
7.4 | IC50 | 15 | Yes | |
KRMLZRDHQHQPJW
|
7.4 | IC50 | 5 | Yes | |
MCIAOHYVDXDCLF
|
7.4 | Ki | 8 | Yes | |
AMSOPBXQXSAAAC
|
7.4 | IC50 | 12 | Yes | |
JHLONFVVTLRHIZ
|
7.4 | IC50 | 4 | — | |
XYUFCXJZFZPEJD
|
7.4 | IC50 | 3 | — | |
XYUFCXJZFZPEJD
|
7.4 | IC50 | 9 | — | |
XYUFCXJZFZPEJD
|
7.4 | IC50 | 23 | Yes | |
INDMCILJGPHHCG
|
7.4 | Ki | 3 | — | |
MMVHNEPFDQHBTM
|
7.4 | IC50 | 5 | Yes | |
KJGUOQMSLKZPAT
|
7.4 | IC50 | 17 | Yes | |
NTUVEMUMVHHACY
|
7.4 | IC50 | 12 | Yes | |
NXSJMRCTGYTSTK
|
7.4 | Kd | 200 | — | |
ADNDQUKOVGKCGQ
|
7.4 | Ki | 3 | — | |
KDOMXVVBKAYVDL
|
7.4 | Ki | 3 | — | |
RVIJQMOQZFCSHL
|
7.4 | Ki | 8 | Yes | |
CGIUQTLYFGDGTD
|
7.4 | IC50 | 4 | — | |
KOZFSFOOLUUIGY
|
7.3 | IC50 | 88 | Yes | |
OHMCEYCPFVOSNY
|
7.3 | IC50 | 3 | — | |
WKZTVBCDQYBGBO
|
7.3 | IC50 | 16 | Yes | |
LBRQDCWYCRVFAG
|
7.3 | IC50 | 4 | — | |
XYUFCXJZFZPEJD
|
7.3 | IC50 | 6 | — | |
HCJOTKSJPHFVJC
|
7.3 | IC50 | 6 | — | |
IRGJDPZJEUYSKS
|
7.3 | IC50 | 7 | — | |
IRGJDPZJEUYSKS
|
7.3 | IC50 | 9 | — | |
IRGJDPZJEUYSKS
|
7.3 | IC50 | 9 | — | |
IRGJDPZJEUYSKS
|
7.3 | IC50 | 6 | — | |
IVGCXWIFBNPPBW
|
7.3 | IC50 | 6 | — | |
MDHNNGDJYHAYKJ
|
7.3 | IC50 | 12 | Yes | |
USEYXZSHZLLAJS
|
7.3 | IC50 | 6 | — | |
VEMLCWMDXJGJLI
|
7.3 | Ki | 8 | Yes | |
LTGPAFCQBMWTBC
|
7.3 | IC50 | 5 | Yes |