Target Details
| UniProt AC | Q02156 |
|---|---|
| Gene Symbol | PRKCE |
| Protein Name | Protein kinase C epsilon type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 423
- Clinical molecules 146
- Avg pChEMBL 7.28
KEGG Pathways (13)
- AGE-RAGE signaling pathway in diabetic complications
- Aldosterone synthesis and secretion
- Apelin signaling pathway
- Fc gamma R-mediated phagocytosis
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- MicroRNAs in cancer
- Shigellosis
- Sphingolipid signaling pathway
- Tight junction
- Type II diabetes mellitus
- Vascular smooth muscle contraction
- cGMP-PKG signaling pathway
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KAJIDAUQCMSGGN
|
7.8 | IC50 | 8 | Yes | |
SMZYTCQRZVNFFJ
|
7.8 | IC50 | 16 | Yes | |
DDBJOZVQHUZKJJ
|
7.8 | Ki | 4 | — | |
OSVUGUHRKMMBSE
|
7.8 | Kd | 170 | — | |
YIZRPXUMLQCIMQ
|
7.8 | IC50 | 9 | — | |
YRYJOPMCJLSMNU
|
7.8 | IC50 | 6 | — | |
JFAIQUNDRVEIFN
|
7.8 | Ki | 2 | — | |
CIVFNZIOXQANAM
|
7.8 | IC50 | 5 | — | |
CXSQMXRQOZZFLD
|
7.8 | IC50 | 18 | — | |
MODWLWDUUDGOEB
|
7.8 | IC50 | 5 | Yes | |
NSAORZLENDLHHH
|
7.8 | Ki | 2 | — | |
PBCZSGKMGDDXIJ
|
7.8 | IC50 | 68 | Yes | |
QJVMNACFDUTHPM
|
7.8 | IC50 | 6 | — | |
CSCOHEYTBLBQMG
|
7.8 | IC50 | 7 | Yes | |
LPMWTDXPUOFZOV
|
7.8 | Ki | 7 | — | |
XWKJUHBICAMYNW
|
7.8 | Ki | 6 | — | |
FXGHOAZJQNLNFD
|
7.8 | IC50 | 13 | Yes | |
IHPBZPYDPATSLB
|
7.8 | Ki | 2 | — | |
MIUMXIIYGOSUSN
|
7.7 | Ki | 3 | — | |
OQICVMYHDNIADM
|
7.7 | IC50 | 6 | — | |
RSTWARDIGORXQU
|
7.7 | Ki | 7 | Yes | |
SMOYJWUKHYTHIN
|
7.7 | Ki | 2 | — | |
WNDOFCPEDZYDPL
|
7.7 | IC50 | 10 | — | |
AQGHYUYFBXMRBC
|
7.7 | IC50 | 6 | — | |
GRAHICROOXJIEL
|
7.7 | Ki | 3 | — | |
IDSZLHFEKAUIOL
|
7.7 | IC50 | 7 | Yes | |
TUTVKAOMRMMGTD
|
7.7 | Ki | 3 | — | |
AZIMEXGKUWHPQV
|
7.7 | IC50 | 12 | Yes | |
FSBMWCWKNXQVMP
|
7.7 | IC50 | 12 | Yes | |
MKPSMRQVGPTYRL
|
7.7 | IC50 | 6 | — | |
YUKJJLKBBAFYNN
|
7.7 | IC50 | 12 | Yes | |
XSHQBIXMLULFEV
|
7.7 | IC50 | 13 | — | |
XYUFCXJZFZPEJD
|
7.7 | IC50 | 9 | — | |
AJTSZCJSPWNPKP
|
7.6 | Ki | 2 | — | |
GQLCVGQQDYKVCM
|
7.6 | Ki | 2 | — | |
UIZGGLNYSWRCAR
|
7.6 | Ki | 2 | — | |
UWDSNDOLVCLEJW
|
7.6 | Ki | 8 | Yes | |
AJFLRCLZEMUXCH
|
7.6 | IC50 | 4 | — | |
LLEJIEBFSOEYIV
|
7.6 | IC50 | 4 | — | |
OWLWQUHZHTVSAN
|
7.6 | IC50 | 6 | — | |
WQEXBJWFPAMSGJ
|
7.6 | Ki | 8 | Yes | |
UIZGGLNYSWRCAR
|
7.6 | Ki | 2 | — | |
JSXUDEUMWQFINT
|
7.6 | Ki | 3 | — | |
KPCVAMMFCPIUIU
|
7.5 | IC50 | 12 | Yes | |
MVPSDKPPZLPMBB
|
7.5 | Ki | 7 | Yes | |
QEPARSUKSLKMMO
|
7.5 | IC50 | 7 | Yes | |
BPNNZZBLGSVSAA
|
7.5 | IC50 | 6 | — | |
BPNNZZBLGSVSAA
|
7.5 | IC50 | 7 | — | |
BPNNZZBLGSVSAA
|
7.5 | IC50 | 6 | — | |
BPNNZZBLGSVSAA
|
7.5 | IC50 | 7 | — |