Target Details
| UniProt AC | Q02156 |
|---|---|
| Gene Symbol | PRKCE |
| Protein Name | Protein kinase C epsilon type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 423
- Clinical molecules 146
- Avg pChEMBL 7.28
KEGG Pathways (13)
- AGE-RAGE signaling pathway in diabetic complications
- Aldosterone synthesis and secretion
- Apelin signaling pathway
- Fc gamma R-mediated phagocytosis
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- MicroRNAs in cancer
- Shigellosis
- Sphingolipid signaling pathway
- Tight junction
- Type II diabetes mellitus
- Vascular smooth muscle contraction
- cGMP-PKG signaling pathway
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QVOXHUHSSXCOAL
|
8.2 | Ki | 2 | — | |
OAVGBZOFDPFGPJ
|
8.2 | IC50 | 42 | Yes | |
UYBWOWHCXDBQRO
|
8.2 | IC50 | 6 | — | |
SAYMBMAHSBYKKR
|
8.2 | IC50 | 12 | Yes | |
NAQPRTABUZMXQG
|
8.2 | Ki | 3 | — | |
SZJIXBKHTOPEKG
|
8.2 | IC50 | 6 | Yes | |
NSAORZLENDLHHH
|
8.2 | Ki | 2 | — | |
KQEBVHBFIFTJGM
|
8.2 | Ki | 3 | — | |
QUTRNEOYUSHTBW
|
8.2 | Ki | 3 | — | |
TUKOILYAIRACKC
|
8.2 | IC50 | 7 | Yes | |
VANSLOBMJZSUSD
|
8.2 | Ki | 2 | — | |
VLUGUCDUHZVABE
|
8.2 | IC50 | 6 | — | |
LUZOFMGZMUZSSK
|
8.1 | Ki | 8 | Yes | |
GVSRILDMSGVJTR
|
8.1 | IC50 | 7 | — | |
KHGDEZDNICAMOO
|
8.1 | IC50 | 6 | — | |
XTCHBPCWJUSYFA
|
8.1 | IC50 | 5 | Yes | |
FKPDQMIETMHJBH
|
8.1 | Ki | 4 | — | |
XELZELDAOXMYOD
|
8.1 | Ki | 3 | — | |
AJTSZCJSPWNPKP
|
8.1 | Ki | 2 | — | |
MFAQYJIYDMLAIM
|
8.1 | Kd | 130 | Yes | |
POTTVLREWUNNRO
|
8.1 | IC50 | 17 | Yes | |
QMGUOJYZJKLOLH
|
8.1 | IC50 | 21 | Yes | |
CKCJAVJYEBDBEI
|
8.0 | Ki | 5 | — | |
PGBOLFMQGRFIRL
|
8.0 | Ki | 5 | — | |
DXZRDTKQTWORHB
|
8.0 | Ki | 3 | — | |
ZRYGSUWUNVQPFR
|
8.0 | IC50 | 6 | — | |
CDXNZQYZADSNCP
|
8.0 | IC50 | 12 | Yes | |
DDHFNAASWMLNPJ
|
8.0 | Ki | 3 | — | |
DSXXEELGXBCYNQ
|
8.0 | IC50 | 28 | Yes | |
FCVHMDURXUOCFY
|
8.0 | IC50 | 6 | — | |
FCVHMDURXUOCFY
|
8.0 | IC50 | 7 | — | |
FFKRSNGYONHGEV
|
8.0 | IC50 | 12 | Yes | |
IREQISFDFPAXPP
|
8.0 | IC50 | 2 | — | |
OPQUGNXQOSDRMT
|
8.0 | IC50 | 12 | Yes | |
PGWBJRRPIUVOAD
|
8.0 | IC50 | 12 | Yes | |
YIZRPXUMLQCIMQ
|
8.0 | IC50 | 7 | — | |
YIZRPXUMLQCIMQ
|
8.0 | IC50 | 9 | — | |
YIZRPXUMLQCIMQ
|
8.0 | IC50 | 6 | — | |
IHPBZPYDPATSLB
|
8.0 | Ki | 2 | — | |
BPNUQXPIQBZCMR
|
8.0 | Kd | 83 | Yes | |
JHFLXYPDFJHPMX
|
8.0 | IC50 | 6 | — | |
IPBIYLHQBHMHCN
|
7.9 | Ki | 2 | — | |
OLTHFAIHFDAJGG
|
7.9 | IC50 | 5 | Yes | |
ZETICKHKBWHSEB
|
7.9 | Ki | 4 | — | |
XELZELDAOXMYOD
|
7.9 | Ki | 3 | — | |
PBCZSGKMGDDXIJ
|
7.9 | IC50 | 14 | Yes | |
QYTBMLLWBZLPMF
|
7.9 | IC50 | 6 | — | |
PQLKHTRGIRKEMK
|
7.9 | Ki | 3 | — | |
GPGZMTPPOHCJRE
|
7.8 | IC50 | 16 | Yes | |
GQLCVGQQDYKVCM
|
7.8 | Ki | 2 | — |