Target Details
| UniProt AC | Q02156 |
|---|---|
| Gene Symbol | PRKCE |
| Protein Name | Protein kinase C epsilon type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00168 (C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 423
- Clinical molecules 146
- Avg pChEMBL 7.28
KEGG Pathways (13)
- AGE-RAGE signaling pathway in diabetic complications
- Aldosterone synthesis and secretion
- Apelin signaling pathway
- Fc gamma R-mediated phagocytosis
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- MicroRNAs in cancer
- Shigellosis
- Sphingolipid signaling pathway
- Tight junction
- Type II diabetes mellitus
- Vascular smooth muscle contraction
- cGMP-PKG signaling pathway
Active Molecules (423)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WTXAWDOYPWWUJL
|
10.1 | IC50 | 11 | — | |
SSXCVTWCXHGTLK
|
9.9 | IC50 | 11 | — | |
KTGVSZYYHHRRGW
|
9.8 | IC50 | 11 | — | |
VIESIZQAHOPEBR
|
9.8 | IC50 | 11 | — | |
FCYKUTUWVZTVAK
|
9.8 | Kd | 4 | — | |
NVYBXIDWOJVGQI
|
9.8 | IC50 | 11 | — | |
APVOCXHEVZBCGS
|
9.7 | IC50 | 11 | — | |
BQJRUJTZSGYBEZ
|
9.7 | Kd | 4 | — | |
DHTLXMRCLSUJPP
|
9.7 | IC50 | 11 | — | |
MJQUEDHRCUIRLF
|
9.6 | Kd | 4 | — | |
HKSZLNNOFSGOKW
|
9.6 | Kd | 213 | — | |
VVRRZOFLLJAMIK
|
9.4 | IC50 | 11 | — | |
PHEDXBVPIONUQT
|
9.3 | Ki | 6 | Yes | |
QZVQSVZEEJEZSI
|
9.3 | Kd | 5 | — | |
DASVAQCTVIQROX
|
9.3 | Ki | 8 | Yes | |
REAZZDPREXHWNV
|
9.2 | Ki | 7 | — | |
FANQQVWXAKUWNI
|
9.2 | IC50 | 6 | — | |
BQJRUJTZSGYBEZ
|
9.1 | Kd | 13 | Yes | |
WAKGEHXTOOFEAE
|
9.1 | IC50 | 27 | — | |
HXWARSZQGAFXJM
|
9.0 | Ki | 7 | — | |
SUQYTYOVPXAUGB
|
9.0 | Ki | 5 | — | |
HKSZLNNOFSGOKW
|
8.9 | IC50 | 49 | Yes | |
RHJPBGWFGOAEID
|
8.9 | Ki | 8 | Yes | |
XSJFPSCYMJFDNI
|
8.9 | Ki | 7 | — | |
XKEOGEXDEKIDNA
|
8.8 | Ki | 3 | — | |
GMQQMSKNSNVPOW
|
8.8 | IC50 | 9 | Yes | |
QZCYXWFWSDBJGL
|
8.8 | Ki | 8 | Yes | |
NVSJOASGKCGXBZ
|
8.8 | IC50 | 16 | Yes | |
QVOXHUHSSXCOAL
|
8.7 | Ki | 2 | — | |
QYBVZIIWBRIXMX
|
8.7 | IC50 | 12 | Yes | |
RDFXBYJUHGEYHA
|
8.7 | IC50 | 9 | Yes | |
SWKUTOXEFLDOID
|
8.7 | Ki | 7 | — | |
UZCZCOMLMMSRLY
|
8.7 | IC50 | 6 | — | |
JZLFYMHIISZQCZ
|
8.7 | IC50 | 12 | Yes | |
YHESSERBDSKRDZ
|
8.7 | Ki | 4 | — | |
BUCGAQTZOOCIRW
|
8.6 | IC50 | 5 | Yes | |
DZIUPOCVDSYPSY
|
8.6 | IC50 | 8 | Yes | |
NMMBOAVVJDOKHT
|
8.6 | Ki | 3 | — | |
XXJXHXJWQSCNPX
|
8.5 | IC50 | 7 | — | |
URLJNGHIJZMXTK
|
8.4 | IC50 | 6 | — | |
ZOLWRJUQMXEKEO
|
8.4 | IC50 | 6 | — | |
KMFOKKGKNMQAAN
|
8.4 | IC50 | 6 | — | |
VDBJPTBJJMQNOW
|
8.4 | IC50 | 6 | — | |
VANSLOBMJZSUSD
|
8.3 | Ki | 2 | — | |
OBRQLJITIRIMLQ
|
8.3 | IC50 | 11 | — | |
YUJAAMQBNNAQRP
|
8.3 | IC50 | 6 | — | |
JFAIQUNDRVEIFN
|
8.3 | Ki | 2 | — | |
KGPGFQWBCSZGEL
|
8.3 | Kd | 59 | Yes | |
CVCIQKJLZNEUAZ
|
8.3 | IC50 | 7 | Yes | |
HKSZLNNOFSGOKW
|
8.2 | IC50 | 408 | — |