Target Details
UniProt ACQ01726
Gene SymbolMC1R
Protein NameMelanocyte-stimulating hormone receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 516
  • Clinical molecules 0
  • Avg pChEMBL 7.73
Associated Diseases (2)
Top Co-occurrence Targets
Active Molecules (516)
InChIKey pChEMBL Type Targets Clinical
GSOVKXCTSWIFEY 6.6 Ki 2
IGSPGKUFVFMXQE 6.6 Ki 2
WZIILWAZGXRRFZ 6.6 IC50 2
YWRRNKAZKAJGFT 6.6 Ki 2
BEGFBZSFSWOZDK 6.6 Ki 4
HGBJQFBJSTUQOF 6.6 Ki 3
JICSVJQEGDFDBH 6.6 Ki 3
KYLMYZLCQJJVMF 6.6 IC50 4
JPRKCJZGKZFHOW 6.5 IC50 3
MSRUJRYKGIBVTG 6.5 IC50 4
YPCZQXKWTSFFSU 6.5 Ki 2
ZLLOVWBBACAVIV 6.5 Ki 3
ALUGMAFCICEWDO 6.5 IC50 3
DEKJJIFFJPAHRM 6.5 IC50 2
FFAUSQSMDWHWML 6.5 Ki 2
FVGGQGIVDDOMKK 6.5 Ki 2
HLCHESOMJVGDSJ 6.5 Ki 4
PGJYWMVUWDKZMU 6.5 IC50 2
RQHOEQDAYOKRHG 6.5 Ki 3
AIVKUJJDLDHLNN 6.5 Ki 3
YSZTVMQFORZYJG 6.5 IC50 4
FJGOVJXGOUSTAU 6.5 Ki 2
DBZMYFPVMVRJJO 6.5 Ki 2
DXKQQTYKXIZRRJ 6.5 Ki 2
VJXLJBSRIOMQLS 6.5 IC50 4
KWPBFXVTEVUNPD 6.5 IC50 4
BACKPKKWDGBCRT 6.4 Ki 3
LKFLMXAGXFBGSV 6.4 Ki 3
MSXFGNGAAAPRSR 6.4 Ki 3
NDRYSEKKAUQGGO 6.4 IC50 3
NSBYFZXDVSHNEF 6.4 Ki 3
NVXVBSBXBTZZNU 6.4 Ki 3
AWKJUBFDTQDCHX 6.4 Ki 2
DNYQDGRNDXYRDY 6.4 Ki 2
UHAQQQFLDCOOEA 6.4 Ki 2
ZPOQUKYSTRZAFA 6.4 Ki 2
BXJJBQWOZVLBPK 6.4 IC50 3
AODONYDDQNDROG 6.4 IC50 2
JGBGNKDRAKSUHZ 6.4 Ki 4
OFPOZEFXTIZAHE 6.4 Ki 4
XGLWBUKNYXLAFF 6.4 Ki 2
YEXGHTGVNJDCFJ 6.4 Ki 3
VWRQHODLDKRSNP 6.4 IC50 4
XFRXFJPUAKFDHC 6.4 Ki 2
WUDKHRNOVXFNLO 6.4 Ki 2
HIGBPTITEJOMDX 6.4 Ki 2
KCCNZMWUXYDOPS 6.4 IC50 2
SSOJHWGDEMWTNO 6.4 Ki 2
JMNUTDPHHUFMOG 6.4 Ki 4
VILSSUAARNTCPC 6.4 IC50 3
2D structure