Target Details
UniProt ACQ01726
Gene SymbolMC1R
Protein NameMelanocyte-stimulating hormone receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 516
  • Clinical molecules 0
  • Avg pChEMBL 7.73
Associated Diseases (2)
Top Co-occurrence Targets
Active Molecules (516)
InChIKey pChEMBL Type Targets Clinical
DUSMRMPLECSLRG 6.8 Ki 3
RZFOKMNOCAQLCI 6.8 Ki 2
ZZZCDEAVWIKQBQ 6.8 Ki 2
FEKXKTLLBDRSQH 6.8 Ki 2
ROTIMMRQYLIORG 6.8 Ki 2
WLIRRQCYHFOXGC 6.8 IC50 4
GCCDXQSIABULHP 6.8 IC50 3
HYNXKHHGAXLIEQ 6.8 Ki 3
JOWUFLPXVQKTNW 6.8 Ki 3
QHXULIILOQCKTQ 6.8 IC50 3
REGPMQLCJMICLA 6.8 Ki 2
NPVNOTIZHSHLKZ 6.8 Ki 3
VVUGZLZXEFCSGI 6.8 Ki 2
RDQOUEKWQGRDRJ 6.8 Ki 3
UDIAMBWWCWFAJW 6.8 IC50 3
UYKWHGIEHONMDL 6.8 IC50 4
PRPVNAJQUHNHLC 6.8 IC50 3
CGKDFZAWOUIFNO 6.7 Ki 3
JMAZWXVWUNQOOV 6.7 Ki 3
QEQUHVRIJFFOKD 6.7 IC50 4
XOJTYHDBHOXJDL 6.7 IC50 3
NMMRTJBOGUWCEQ 6.7 Ki 4
PQOAIQOLRRUAHF 6.7 Ki 2
QTGLDSNZORTQEK 6.7 IC50 4
VNTJATGNGDRIFN 6.7 IC50 2
ZSWPGAPVLVMTJG 6.7 Ki 2
CQUKLRIOLMQYDE 6.7 IC50 4
SGKSNHUSKUVYHG 6.7 Ki 2
SGKSNHUSKUVYHG 6.7 Ki 2
SYYCZXDFWBANLC 6.7 Ki 3
LMTCYYTZYVZVDJ 6.7 Ki 4
SOCBNUUFEBTEOP 6.7 IC50 3
SOCBNUUFEBTEOP 6.7 IC50 3
ORPYCWJPNJKZIA 6.7 IC50 4
QECOLCQUUXFPQQ 6.7 Ki 2
WOWDZBDFXRWMIV 6.7 Ki 3
RBKDACLJKAMLFN 6.6 IC50 3
SAYNLXAIIPDZPE 6.6 IC50 2
SNEMRJZDOOLWPZ 6.6 Ki 4
MMBHRGOCQSTXRS 6.6 Ki 2
GTMASPVXPKDKOK 6.6 Ki 3
WCVJJQCPIDBNFM 6.6 IC50 4
YUKODIVVRQEHLF 6.6 IC50 3
GVUXGBSAZGMQMX 6.6 Ki 2
ONWSRSOVEDSAJV 6.6 IC50 4
UAISFSHHKXHKOI 6.6 IC50 4
MWOCTFMMKHRPCY 6.6 IC50 2
DCOSVJTYYUGOGC 6.6 Ki 2
KOMGNGDDTPNSKC 6.6 Ki 3
YENCSZMEVJAKQJ 6.6 IC50 4
2D structure