Target Details
UniProt ACQ01726
Gene SymbolMC1R
Protein NameMelanocyte-stimulating hormone receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 516
  • Clinical molecules 0
  • Avg pChEMBL 7.73
Associated Diseases (2)
Top Co-occurrence Targets
Active Molecules (516)
InChIKey pChEMBL Type Targets Clinical
HDBFFTYMERRCIX 8.0 IC50 3
UNXFCHHFXJFRRB 8.0 Ki 3
RUDWSQPLBXOLBE 8.0 IC50 3
GZWUQPQBOGLSIM 8.0 IC50 4
XVPBPJWOKGRCPR 7.9 Ki 3
BPRBXYIGPSSVII 7.9 Ki 2
LICCWOCOLMEXQP 7.9 Ki 4
MZFOEDJULWOZIV 7.9 IC50 3
KZXNIFOXWZLCOK 7.9 IC50 4
FRLGHEFWPNKBDQ 7.9 Ki 2
KXPKJVIQPPHENQ 7.9 Ki 2
CFAHIOAXVOKBCK 7.9 IC50 3
AXYNQPYLILCAPC 7.8 Ki 3
CBZNNNCTDMTAGU 7.8 Ki 3
DNDWQJKQEQLRTQ 7.8 Ki 3
OHFHKCOOPQLGKC 7.8 Ki 3
VSVABBLUDNGFCZ 7.8 Ki 2
LKGYQUQHVGIHMG 7.8 IC50 3
ASUAOIWGQADQOH 7.8 Ki 3
DOAQTQYFNKQPTO 7.8 IC50 2
SPJYDEIJYHHMBB 7.8 IC50 3
UNXFCHHFXJFRRB 7.8 Ki 3
XMQSVPKHHVWBGS 7.8 IC50 4
DZBWWVGXDVRUHV 7.8 Ki 3
FEKXKTLLBDRSQH 7.8 Ki 3
VLXDEFRTAJLNNA 7.8 Ki 3
YZQBDVJPOXNSJR 7.7 Ki 3
CRWGRYHHKDTXFC 7.7 IC50 3
UICVQJGBBAMKDX 7.7 Ki 4
YQOPVQXIKMEFFV 7.7 IC50 4
YJCDHAJJLSUBDS 7.7 IC50 4
FZMMHTRNAWCOMM 7.7 Ki 3
ROTHBSFMHAHRTG 7.7 IC50 4
LNVJOUMPGCMIDQ 7.7 IC50 3
WZIILWAZGXRRFZ 7.7 IC50 3
NIGXYCDFYWYVQS 7.6 Ki 2
XANHKAKFNIWYOE 7.6 IC50 4
CVFGCUVAZVPTRO 7.6 IC50 2
ANTVHWLGFDSXEN 7.6 Ki 2
OLKZRPFXLZQEOU 7.6 Ki 2
MJWHBKTUULEGMJ 7.6 Ki 3
UIMWAMYMWYXGRV 7.5 Ki 2
GGYWLZFXFKFWKL 7.5 IC50 4
DBJGVYJTQHCOAH 7.5 Ki 2
KXJHWAIMDKIUMK 7.5 Ki 2
PJDCKQFLLOIVHJ 7.5 Ki 3
XTGXCCGBTWVVAZ 7.5 Ki 3
ZKTNTRAJYNNFHC 7.5 Ki 3
SHUMMQAOTPBZAQ 7.5 Ki 2
RQIFYTAAHPOYSP 7.5 Ki 3
2D structure