Target Details
UniProt ACQ01726
Gene SymbolMC1R
Protein NameMelanocyte-stimulating hormone receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 516
  • Clinical molecules 0
  • Avg pChEMBL 7.73
Associated Diseases (2)
Top Co-occurrence Targets
Active Molecules (516)
InChIKey pChEMBL Type Targets Clinical
SVSUFMZEUZIVDX 8.5 Ki 2
QOZPHXSKYHWXNY 8.5 IC50 4
RQZHKEFEFWSLOK 8.5 Ki 3
UBKGFMZTCLCOLM 8.5 Ki 4
DZOXHHUQYQUKJB 8.5 Ki 4
RHDRZFXISWDZNM 8.5 Ki 3
AUPOJQYWSLXSAP 8.5 Ki 3
YBWGYSWBATYFBD 8.5 IC50 4
GVLRCXVPKHTHFV 8.4 Ki 3
KXWAHHUIDLURNT 8.4 Ki 4
IVQPGYKGSXUDKV 8.4 IC50 4
IXLVDOBKTIIMBE 8.4 Ki 4
XQQIIPUPHPWBDF 8.4 Ki 3
DLVAKQPHOINITK 8.4 IC50 4
WQIHSOXKRYCWEW 8.4 Ki 4
KPKOJXZVOJTTBP 8.4 IC50 2
PCKSOAZIMLQBHU 8.4 Ki 4
WSLQGTFNIJDQNS 8.4 Ki 2
DQDUAZXNONBSMT 8.4 Ki 3
BZEWEHPSOMSRJV 8.4 Ki 3
HDHDTKMUACZDAA 8.3 Ki 3
PIVHBXZYYYPXHW 8.3 IC50 4
VNKGTZHAAMHYKK 8.3 Ki 3
WRKBOTGDFLBBDK 8.3 Ki 2
YBKZXQIAHZXKIW 8.3 Ki 3
HNVXASMBDVOKKN 8.3 IC50 3
AOMUTEUZPCRNFD 8.2 Ki 3
TWDTYJMEGITLBP 8.2 IC50 3
OBKWMOSDTIUARN 8.2 Ki 2
PPISUPSPKCHLKT 8.2 Ki 3
WHNFPRLDDSXQCL 8.2 IC50 4
ZJRYSELENYTFKR 8.2 Ki 3
ZTSQVRSYAGAZPG 8.2 IC50 4
VIJAYCRGMXEAAI 8.2 Ki 3
UYOAPGITMAMCFT 8.1 IC50 4
KRKYTJXTDCSSJS 8.1 IC50 4
OGIIVLJDBHLNNQ 8.1 Ki 2
XTFWFFODDNNYFQ 8.1 Ki 4
HJMAXNXTRYYRCZ 8.1 Ki 4
KIFNALNSUOJQPJ 8.1 Ki 4
IXQMIHWLSWEYPU 8.1 IC50 4
UNUGBHUNONVSEZ 8.1 Ki 2
VXVQZXYFPLAEJW 8.1 Ki 3
YAVZBTAEIGLTOG 8.1 Ki 3
JBPCVEBLPIKYKT 8.0 IC50 3
RVVLJWZWXHPMLS 8.0 IC50 4
VHZUXXIKZIQBLB 8.0 Ki 2
PNUQGRIALHGKEH 8.0 Ki 3
QAXKNGODUAVCKD 8.0 Ki 4
CHBTZNAADZTZLP 8.0 Ki 4
2D structure