Target Details
UniProt ACQ01726
Gene SymbolMC1R
Protein NameMelanocyte-stimulating hormone receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 516
  • Clinical molecules 0
  • Avg pChEMBL 7.73
Associated Diseases (2)
Top Co-occurrence Targets
Active Molecules (516)
InChIKey pChEMBL Type Targets Clinical
UMHVNRYGRKBTCG 9.0 IC50 4
CDHOQEHTFUNKKJ 8.9 Ki 3
SFVVQRJOGUKCEG 8.9 Ki 3
FEFWDDKHEOVPCG 8.9 IC50 4
REMHNXQVRVXAGT 8.9 IC50 4
MTFOEQYGYVFQPJ 8.9 Ki 3
HJERQRDKWIWHPW 8.9 Ki 4
NSMUITYTUDRYSP 8.9 Ki 3
QDYYRHYWJPWOTC 8.9 Ki 2
QXRXXIKAVZAGHZ 8.9 IC50 3
UHOVQNZJYSORNB 8.9 Ki 8
UBWLAYRWNUNYHG 8.8 IC50 4
UVJBRYNBZSRMBZ 8.8 Ki 4
DIWJBUBBVDFSOS 8.8 IC50 3
RCULCPVSLOFQPR 8.8 Ki 4
UELLOIOSXYBLCZ 8.8 Ki 3
WHNFPRLDDSXQCL 8.8 IC50 4
FIPGSBWOMGALGM 8.8 Ki 4
JTEJZABLGYDSAQ 8.8 IC50 3
HRTHPANNFOMYJE 8.8 Ki 4
ANGMCMXZFGHVPX 8.7 Ki 3
UAHFGYDRQSXQEB 8.7 Ki 3
YMCLJESYNLOGEG 8.7 Ki 2
YMCLJESYNLOGEG 8.7 Ki 2
FFHBJDQSGDNCIV 8.7 Ki 4
VVNAQHKXBHSZIX 8.7 IC50 3
AWOIGQXOOIHLJT 8.7 Ki 2
KOWZSZLHPBJHEB 8.7 Ki 3
RNCVEEUMKRRHLC 8.7 IC50 4
UKMQKNTZNHDSPD 8.7 IC50 4
WOQVIKOQMYEYTM 8.7 Ki 2
WSDYWWDQJYPQDS 8.7 Ki 3
ZRHYLFBORVIBEU 8.7 Ki 3
HICQRDPLMADMBD 8.7 Ki 4
ULKFOTUQRDIPQX 8.7 Ki 4
KBLNYXZHILRCGF 8.7 Ki 4
QXRXXIKAVZAGHZ 8.7 IC50 2
REMHNXQVRVXAGT 8.6 IC50 4
DIWJBUBBVDFSOS 8.6 IC50 3
IDLFZVILOHSSID 8.6 Ki 3
SSZDAFBCWHVROA 8.6 Ki 3
FDPBRBMLLVILMV 8.6 Ki 3
PWVUYOZSIWYFJW 8.6 Ki 4
SLEIICTWQFRIFM 8.6 Ki 3
UMHVNRYGRKBTCG 8.6 IC50 4
DPPBMHXXQRAKPB 8.6 Ki 4
QCXXYYAQEUNASC 8.6 Ki 3
BCYYSNXZIDIGEG 8.5 Ki 2
FWYIDGAEHPOSEJ 8.5 Ki 2
JQDBJPQYLBLUNL 8.5 Ki 2
2D structure