Target Details
UniProt ACQ01726
Gene SymbolMC1R
Protein NameMelanocyte-stimulating hormone receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 516
  • Clinical molecules 0
  • Avg pChEMBL 7.73
Associated Diseases (2)
Top Co-occurrence Targets
Active Molecules (516)
InChIKey pChEMBL Type Targets Clinical
JDKLPDJLXHXHNV 9.6 IC50 4
OKHXBJLIBJDJMV 9.5 IC50 4
WPNVZVWZWSOGOI 9.5 Ki 2
WSDYWWDQJYPQDS 9.5 IC50 4
AXBBCWVVFWOKFH 9.5 Ki 2
NPGINHVVWSGMMV 9.5 Ki 2
WZIILWAZGXRRFZ 9.5 IC50 4
FJSKRKLUQFIKJP 9.4 Ki 3
PZVZJDCUPVOTTP 9.4 IC50 4
NOLFWMRTIVNJFP 9.4 Ki 4
JLMVHMLMBIPZSW 9.4 Ki 4
JXWMBIOMMZLSIR 9.3 Ki 2
KPFZSXDUVZTNAQ 9.3 IC50 3
CNWHTMNTHKVVEV 9.3 Ki 2
JPHOERRRWXXXOC 9.3 Ki 2
QBYHLGIJWBFDGJ 9.3 IC50 4
RVKSMTBVJXMWFD 9.3 IC50 4
UAHFGYDRQSXQEB 9.3 Ki 5
XQMPAWYRHAOJTE 9.3 Ki 4
IJVUOKFOZUYPMK 9.3 Ki 2
PPKIGEMCDOLKEY 9.2 Ki 3
PPKIGEMCDOLKEY 9.2 Ki 3
WBTHAPYEEKFPSX 9.2 Ki 4
JJRDXXQLVRWOCP 9.2 Ki 2
NSMUITYTUDRYSP 9.2 Ki 3
APAIPJOPPUMQFD 9.2 Ki 4
CADNRYGCBMLNJN 9.2 Ki 3
FHNLUGMXKXPEFR 9.2 IC50 4
VPWMVGOTLXHAFL 9.2 Ki 2
APHPBWUTFHDTLW 9.1 Ki 4
ZKFHMXVIVJCDFY 9.1 Ki 4
PGHLIJXAFOBIIC 9.1 IC50 2
CSIVLBODDQFIPR 9.1 Ki 2
RDLAZLIJEHHWIX 9.1 Ki 2
CRLGCHNGOJRZNC 9.1 Ki 3
KWTLWMHGSUOSHU 9.1 Ki 4
LEURJYAAAHRVRF 9.1 Ki 2
XLLJFSCSXTYVTN 9.1 Ki 4
KSMXNEYOFKPWFI 9.0 Ki 4
WZIILWAZGXRRFZ 9.0 IC50 4
DLOGSFRUKCUWHC 9.0 Ki 2
FPYYFGFPTJRMBR 9.0 IC50 4
GGYWLZFXFKFWKL 9.0 IC50 4
JWBGVBLXXIKBCO 9.0 Ki 2
KWBYYFKCXHSTPA 9.0 IC50 4
KYOVLZCJSUXUJI 9.0 Ki 3
UCFQPBRLCMKTJY 9.0 Ki 2
ZSAXEKUGMLDFHT 9.0 Ki 3
KNWLOSLCTAQNSO 9.0 Ki 4
OFHSVORZHRSITE 9.0 IC50 2
2D structure