Target Details
UniProt ACQ01726
Gene SymbolMC1R
Protein NameMelanocyte-stimulating hormone receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 516
  • Clinical molecules 0
  • Avg pChEMBL 7.73
Associated Diseases (2)
Top Co-occurrence Targets
Active Molecules (516)
InChIKey pChEMBL Type Targets Clinical
ZSRGOYOFHLLWGA 11.3 Ki 2
CHNMWUKSZIMHIX 11.2 Ki 3
DYLFBHOZQPVNMC 11.0 Ki 2
RDCIPOBDQMOUKD 11.0 IC50 4
SAQQSSWKBKHBIG 11.0 Ki 2
UCISBBYZNLQVGP 11.0 Ki 2
VOSIMUPSRJWOJN 11.0 Ki 2
HYWBNHIBZICAAO 10.8 Ki 2
QQVWMYDNTPWWPW 10.8 Ki 2
QYYSVWQCDYOKEJ 10.8 Ki 2
XNPPTTUWPBNRFQ 10.8 Ki 2
UCISBBYZNLQVGP 10.7 Ki 2
KRZXMSMNMZEKGP 10.6 Ki 4
CAXNNMYXBQZZIP 10.6 Ki 2
DVRRTOIJYURKKI 10.6 Ki 2
ZOFPYCCSYGWTCN 10.6 Ki 2
QXEWYZXRQRSHMR 10.5 Ki 2
UNGLYFOZRWHRKE 10.5 Ki 2
MBBQINYFFIKILA 10.5 Ki 3
CATZYTHJWOAGOB 10.4 Ki 2
KPDWCDURFGPKLY 10.4 Ki 2
PYANSLUAUZKUFT 10.4 Ki 2
VGBVAARMQYYITG 10.4 Ki 3
NVIBFTUPAARCBA 10.3 Kd 3
NYBMXOVCJILSIJ 10.3 Ki 2
YXIBEMYOGWJEQC 10.2 Ki 4
YZJAIULMUUQAPH 10.2 Ki 2
PVVLKBSYHAGXBD 10.2 Ki 4
MLXMTZDTPIINBF 10.2 Ki 2
KLOVFBFHFHKKJQ 10.1 IC50 3
XDLJELQQEILLFZ 10.1 Ki 4
BUVGQEXSQXRZQG 10.0 Ki 4
ZSRGOYOFHLLWGA 10.0 Ki 2
KRZXMSMNMZEKGP 10.0 Ki 3
JUOGFOXGQYCMTJ 9.9 Ki 2
KLOVFBFHFHKKJQ 9.9 IC50 3
VDHCRROJIVFVLM 9.8 Ki 4
UWUHDNLMNSCQPX 9.8 Ki 2
IJVUOKFOZUYPMK 9.8 Ki 2
OHFMRHZLQMSCRN 9.8 IC50 4
CHNMWUKSZIMHIX 9.8 Ki 3
AXBBCWVVFWOKFH 9.7 Ki 2
DPJAKAHREXIEPH 9.7 IC50 3
GGYWLZFXFKFWKL 9.7 IC50 3
VSGQPYQAGHZCFG 9.7 Ki 2
ZPANOUCVWZTSLE 9.7 IC50 4
ZSONGANRJTVTCP 9.7 Ki 4
QIKIYIZHGOCQOO 9.6 Ki 3
PHHQWWPLQKXGDH 9.6 Ki 4
HOWXKXAJVJPQOI 9.6 IC50 3
2D structure