Target Details
| UniProt AC | Q01118 |
|---|---|
| Gene Symbol | SCN7A |
| Protein Name | Sodium channel protein type 7 subunit alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00520 (Ion_trans) PF24609 (IQ_SCN5A_C) PF06512 (Na_trans_assoc) |
Summary
- Multi-target molecules 41
- Clinical molecules 0
- Avg pChEMBL 7.69
KEGG Pathways (1)
Active Molecules (41)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WSPHMGORSRQULF
|
11.0 | IC50 | 6 | — | |
GFDXIUXAFNREKM
|
9.2 | IC50 | 6 | — | |
PTCBNPULJWGSML
|
9.2 | IC50 | 9 | — | |
XOAUGYVLRSCGBG
|
9.1 | IC50 | 8 | — | |
DFBDAHMZXJYZJG
|
9.1 | IC50 | 7 | — | |
SXOAHIZWCZOILH
|
8.7 | IC50 | 9 | — | |
TVQFYGIEBVVYRN
|
8.7 | IC50 | 4 | — | |
HXQNEKJQBGXFAG
|
8.5 | IC50 | 2 | — | |
KYBPOTYVFWNSGS
|
8.5 | Kd | 8 | — | |
VENWKQHIOIEAII
|
8.4 | IC50 | 3 | — | |
KWAURGCHFYCYPQ
|
8.3 | IC50 | 4 | — | |
FQHDBBOTIYOYLF
|
8.2 | IC50 | 3 | — | |
SXOAHIZWCZOILH
|
8.1 | IC50 | 3 | — | |
QJETWCFGSMIKHY
|
8.0 | IC50 | 2 | — | |
ZYSCOUXLBXGGIM
|
8.0 | IC50 | 9 | — | |
KSBYUWHBUZLDDL
|
8.0 | IC50 | 2 | — | |
YYVCJPDYCCNDLJ
|
7.9 | IC50 | 2 | — | |
QJNYOQCRJJMAOZ
|
7.8 | IC50 | 3 | — | |
XVGMRZRHSRQQFG
|
7.8 | IC50 | 2 | — | |
DEYOMPPOEBPYPT
|
7.8 | IC50 | 3 | — | |
YKHDDBRKQAIROO
|
7.8 | IC50 | 3 | — | |
SREGSGWKZFYIDY
|
7.7 | IC50 | 3 | — | |
OZPDALRKJRELDR
|
7.7 | IC50 | 2 | — | |
FYMGGEYPNDYSSU
|
7.7 | IC50 | 2 | — | |
KQQXPTRMUYKUIC
|
7.7 | Kd | 8 | — | |
DKLFTDOPHVNBBI
|
7.5 | IC50 | 3 | — | |
CFMYXEVWODSLAX
|
7.4 | IC50 | 8 | — | |
NEBUOXBYNAHKFV
|
7.3 | IC50 | 5 | — | |
YVUQSNJEYSNKRX
|
7.3 | IC50 | 36 | — | |
GKCBAIGFKIBETG
|
7.2 | IC50 | 10 | — | |
KEFLKWVDEZWQCI
|
7.2 | IC50 | 2 | — | |
OZAUCXKCFJDDRB
|
7.1 | IC50 | 2 | — | |
YGCDGFNMFBCJAB
|
6.8 | IC50 | 3 | — | |
RPQXVSUAYFXFJA
|
6.4 | IC50 | 8 | — | |
XYCSIKBESLTOLI
|
6.1 | IC50 | 2 | — | |
REGLDXIVBNZLDY
|
6.1 | IC50 | 2 | — | |
OKFZWUFFIAFNGA
|
6.0 | IC50 | 2 | — | |
BHHALVLOZQTWNJ
|
6.0 | IC50 | 2 | — | |
PSKAASYIVOPYMH
|
6.0 | IC50 | 2 | — | |
HBNPJJILLOYFJU
|
6.0 | IC50 | 21 | — | |
VATOXHDFJPTCPW
|
6.0 | IC50 | 2 | — |