Target Details
| UniProt AC | Q01064 |
|---|---|
| Gene Symbol | PDE1B |
| Protein Name | Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00233 (PDEase_I) PF08499 (PDEase_I_N) |
Summary
- Multi-target molecules 652
- Clinical molecules 0
- Avg pChEMBL 7.96
KEGG Pathways (7)
Active Molecules (652)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TVGMRVMYCDHOEG
|
8.7 | IC50 | 3 | — | |
FDEJYPFAUDLEJD
|
8.6 | IC50 | 3 | — | |
GJZNHSHBNVLOAO
|
8.6 | IC50 | 3 | — | |
AIKXKABMMRXBQU
|
8.6 | IC50 | 3 | — | |
BHFKZPHEMFPTRO
|
8.6 | IC50 | 3 | — | |
FBPBJZZMBZEJSF
|
8.6 | IC50 | 3 | — | |
HCLONMUJAHJFIH
|
8.6 | IC50 | 3 | — | |
JHGCAWXOMLLFMA
|
8.6 | IC50 | 3 | — | |
MLGGVHCQGVZWQR
|
8.6 | IC50 | 3 | — | |
NDQZTZXQHDYXCS
|
8.6 | IC50 | 3 | — | |
PFDYAXRVKURLCH
|
8.6 | IC50 | 3 | — | |
RORWDTCBTBGWNA
|
8.6 | IC50 | 7 | — | |
SDTZIRBETDMBLS
|
8.6 | IC50 | 3 | — | |
SKXWAYULKGVUDE
|
8.6 | IC50 | 3 | — | |
WXGZVKRAYFNMHG
|
8.6 | IC50 | 3 | — | |
YFAHCXPQQYYPCW
|
8.6 | IC50 | 3 | — | |
YGFHMMKTVSGDPM
|
8.6 | IC50 | 3 | — | |
AXEQFCFNPOGNCH
|
8.6 | IC50 | 3 | — | |
IMKYKBMLZRNQRQ
|
8.6 | IC50 | 3 | — | |
BHINMZMKXRIBEG
|
8.6 | IC50 | 3 | — | |
JIGCMFQAIKAHMI
|
8.6 | IC50 | 3 | — | |
SBMPCNJJGZDPRT
|
8.6 | IC50 | 3 | — | |
SJDHGTJKQKPRAR
|
8.6 | IC50 | 3 | — | |
BOOYHBPHFVNWNH
|
8.5 | IC50 | 4 | — | |
DTEHKURDWHCADV
|
8.5 | IC50 | 3 | — | |
MPJXQIBFZBPJFH
|
8.5 | IC50 | 3 | — | |
LYJSPCIIWWKSML
|
8.5 | IC50 | 3 | — | |
OZQQLPFSQLZXQT
|
8.5 | IC50 | 3 | — | |
PZHZVFDPQAUVKV
|
8.5 | IC50 | 3 | — | |
QIWVSVNHRDQBOW
|
8.5 | IC50 | 3 | — | |
XNUXIYGMZDJLFB
|
8.5 | IC50 | 3 | — | |
ZOYWVKURDMXZTC
|
8.5 | IC50 | 3 | — | |
IBAWDCALOOJODQ
|
8.5 | IC50 | 3 | — | |
IRSHUSVLDQPATB
|
8.5 | IC50 | 3 | — | |
POVOCAKFKAXGDL
|
8.5 | IC50 | 3 | — | |
RJISSJINTRICQD
|
8.5 | IC50 | 3 | — | |
CXGJWWJDXYZFFZ
|
8.4 | IC50 | 3 | — | |
ZLTYIDKHKFGNFO
|
8.4 | IC50 | 3 | — | |
HUQJJAUBVULGLS
|
8.4 | IC50 | 3 | — | |
DQKKFAGODSQYOO
|
8.4 | IC50 | 3 | — | |
HINKCAKLUHRIQD
|
8.4 | IC50 | 3 | — | |
ITYGOFCAYSOSFS
|
8.4 | Ki | 2 | — | |
PSUHAEXBWCRQED
|
8.4 | Ki | 2 | — | |
USWMJZZZYCJYJT
|
8.4 | IC50 | 3 | — | |
YKYCEIQQBDUXHL
|
8.4 | IC50 | 3 | — | |
NHHYCGIUZMMXNN
|
8.4 | IC50 | 3 | — | |
YCKJCPNPYHTASY
|
8.4 | IC50 | 3 | — | |
JGQBOOQITKPWJR
|
8.4 | IC50 | 3 | — | |
XIDRGBXOXDHAGV
|
8.4 | IC50 | 3 | — | |
YXBLPELQAKXZRS
|
8.4 | IC50 | 2 | — |