Target Details
| UniProt AC | Q00975 |
|---|---|
| Gene Symbol | CACNA1B |
| Protein Name | Voltage-dependent N-type calcium channel subunit alpha-1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08763 (Ca_chan_IQ) PF16905 (GPHH) PF00520 (Ion_trans) |
Summary
- Multi-target molecules 96
- Clinical molecules 0
- Avg pChEMBL 7.18
KEGG Pathways (15)
- Calcium signaling pathway
- Chemical carcinogenesis - receptor activation
- Cholinergic synapse
- Dopaminergic synapse
- GABAergic synapse
- Huntington disease
- MAPK signaling pathway
- Morphine addiction
- Nicotine addiction
- Pathways of neurodegeneration - multiple diseases
- Prion disease
- Retrograde endocannabinoid signaling
- Serotonergic synapse
- Synaptic vesicle cycle
- Type II diabetes mellitus
Associated Diseases (1)
Active Molecules (96)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RTFHWULQHQDWPK
|
7.0 | IC50 | 26 | — | |
GTSIUFNWVXFHJS
|
7.0 | IC50 | 3 | — | |
AOQSRDPSBXFFQW
|
7.0 | IC50 | 4 | — | |
CEXBUHRJNQKOBZ
|
7.0 | IC50 | 3 | — | |
JDFLEUYRGZPZQD
|
7.0 | IC50 | 3 | — | |
VCPMZDWBEWTGNW
|
7.0 | IC50 | 3 | — | |
AOQSRDPSBXFFQW
|
6.8 | IC50 | 3 | — | |
FMJSSIYEDJFGBC
|
6.8 | IC50 | 3 | — | |
PPVBMJIAJXVQFX
|
6.8 | IC50 | 3 | — | |
POPQMMOUZVBXFY
|
6.8 | IC50 | 3 | — | |
UZBVUMAEAIQRKF
|
6.8 | IC50 | 4 | — | |
JJWWPFHYFYVBMO
|
6.7 | IC50 | 3 | — | |
RPLRXHLXRQIHHQ
|
6.7 | IC50 | 3 | — | |
YYMGRGSETHUACY
|
6.7 | IC50 | 3 | — | |
NKYGAHUSYUIOCV
|
6.7 | IC50 | 2 | — | |
UQEYHZANEBZUSS
|
6.7 | IC50 | 4 | — | |
PSEHTODILBVIHC
|
6.6 | IC50 | 4 | — | |
CBDZLOJIUYHCHO
|
6.6 | IC50 | 4 | — | |
NIMFDABOPDBIHU
|
6.6 | IC50 | 3 | — | |
HWGMUVSZGFXYSD
|
6.6 | IC50 | 3 | — | |
DKVOGZPCCPBBPU
|
6.6 | IC50 | 3 | — | |
QXNYWQVYZYCACA
|
6.6 | IC50 | 3 | — | |
YLVSVJDCTDBERH
|
6.6 | IC50 | 2 | — | |
KGKFKQGQYIUQAL
|
6.6 | IC50 | 3 | — | |
AYURKVVCUVKFLJ
|
6.6 | IC50 | 2 | — | |
DOVZOQYQXHNCCN
|
6.5 | IC50 | 3 | — | |
YZBMBXSAQFTDCP
|
6.5 | IC50 | 3 | — | |
MLTWOMDQQFOCMD
|
6.5 | IC50 | 3 | — | |
PVJNWPXQHNFPOR
|
6.5 | IC50 | 3 | — | |
APFIMMRBLUEEJX
|
6.5 | IC50 | 3 | — | |
NTCNYPJNYIBPSC
|
6.5 | IC50 | 3 | — | |
MTACWCHMAADIEZ
|
6.5 | IC50 | 3 | — | |
QJXZQIYIFNIJIO
|
6.4 | IC50 | 3 | — | |
DXHGSDDDNQXAEJ
|
6.4 | IC50 | 26 | — | |
HBNPJJILLOYFJU
|
6.4 | IC50 | 21 | — | |
SZXAWCKROBFQPN
|
6.3 | IC50 | 3 | — | |
RLEMIIBGFDBVBD
|
6.3 | IC50 | 3 | — | |
GGKXNHJATNHIDB
|
6.3 | IC50 | 3 | — | |
GYDSTQXJLLEDBS
|
6.3 | IC50 | 3 | — | |
RFHHKLHLLXMGOX
|
6.3 | IC50 | 3 | — | |
KGQXWNGARPKIIX
|
6.2 | IC50 | 3 | — | |
KAQSYOBVGLVJFK
|
6.1 | IC50 | 2 | — | |
YZALTYFOCATYBV
|
6.1 | IC50 | 2 | — | |
XKDFZZUFCHOVRN
|
6.1 | IC50 | 27 | — | |
DUTNQEVLPMRTHE
|
6.1 | IC50 | 2 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — |