Target Details
| UniProt AC | Q00613 |
|---|---|
| Gene Symbol | HSF1 |
| Protein Name | Heat shock factor protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00447 (HSF_DNA-bind) PF06546 (Vert_HS_TF) |
Summary
- Multi-target molecules 22
- Clinical molecules 0
- Avg pChEMBL 7.08
KEGG Pathways (1)
Active Molecules (22)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PIMQWRZWLQKKBJ
|
8.2 | IC50 | 36 | — | |
IYYAIKPZMIMDEQ
|
8.1 | IC50 | 2 | — | |
KXBKPNSSZAFEBH
|
7.8 | IC50 | 3 | — | |
CODOEMQMKTTYRW
|
7.8 | IC50 | 7 | — | |
KLHOCHQJHXNKAS
|
7.7 | IC50 | 2 | — | |
RZQWMJAOUJLEAM
|
7.6 | IC50 | 3 | — | |
YTWDOCYUHJCFCG
|
7.5 | IC50 | 3 | — | |
HRGRQFYTVDLKEE
|
7.4 | IC50 | 3 | — | |
JCQSAYNTEFQHGH
|
7.3 | IC50 | 5 | — | |
JCQSAYNTEFQHGH
|
7.3 | IC50 | 3 | — | |
QLQYWGHSSLXLOS
|
7.2 | IC50 | 5 | — | |
CQLFRGIYOHYSJV
|
7.1 | IC50 | 7 | — | |
ORLJHIALWUUFDA
|
6.9 | IC50 | 2 | — | |
VKUXBRRQHBTQPW
|
6.8 | IC50 | 3 | — | |
NYPBFUANCHGSJU
|
6.7 | IC50 | 3 | — | |
LLTXIVYBCVSFHB
|
6.7 | IC50 | 2 | — | |
REJHOMMDDHCCJU
|
6.5 | IC50 | 3 | — | |
AWYBHCVXZFMJHV
|
6.3 | IC50 | 5 | — | |
SDVZKQSDNMFMHZ
|
6.3 | IC50 | 2 | — | |
KWBCXZRKOCGHBO
|
6.2 | IC50 | 3 | — | |
YTFMKHAFPHBMNE
|
6.1 | IC50 | 3 | — | |
UWHMFXHWZZSXIB
|
6.1 | IC50 | 3 | — |