Target Details
| UniProt AC | Q00537 |
|---|---|
| Gene Symbol | CDK17 |
| Protein Name | Cyclin-dependent kinase 17 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 33
- Clinical molecules 9
- Avg pChEMBL 6.96
Active Molecules (33)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JRNJNYBQQYBCLE
|
9.1 | Kd | 40 | Yes | |
OVPNQJVDAFNBDN
|
9.0 | Kd | 44 | Yes | |
ALKJNCZNEOTEMP
|
8.3 | Kd | 55 | — | |
WVXNSAVVKYZVOE
|
8.2 | Kd | 92 | — | |
OUSFTKFNBAZUKL
|
7.9 | Kd | 58 | Yes | |
AYCPARAPKDAOEN
|
7.8 | Kd | 73 | — | |
ODPGGGTTYSGTGO
|
7.8 | Kd | 153 | — | |
HKSZLNNOFSGOKW
|
7.8 | IC50 | 408 | — | |
BFSMGDJOXZAERB
|
7.4 | Kd | 33 | — | |
RPGZQOOZHIEPJW
|
7.2 | Kd | 18 | — | |
RPGZQOOZHIEPJW
|
7.2 | Kd | 18 | — | |
MZDKLVOWGIOKTN
|
7.0 | Kd | 80 | — | |
XZXHXSATPCNXJR
|
7.0 | Kd | 165 | Yes | |
HKSZLNNOFSGOKW
|
7.0 | Kd | 213 | — | |
MWKSRKSEWLRPBL
|
6.9 | Kd | 1075 | — | |
ASUGUQWIHMTFJL
|
6.9 | Kd | 18 | — | |
CXQHYVUVSFXTMY
|
6.8 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.8 | Kd | 149 | — | |
KDKUVYLMPJIGKA
|
6.5 | Kd | 91 | Yes | |
NHHQJBCNYHBUSI
|
6.5 | Kd | 220 | — | |
PHXJVRSECIGDHY
|
6.5 | Kd | 59 | — | |
JOOXLOJCABQBSG
|
6.5 | Kd | 139 | — | |
LNMRSSIMGCDUTP
|
6.4 | Kd | 13 | — | |
BIIVYFLTOXDAOV
|
6.3 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
6.3 | Kd | 82 | Yes | |
FNHKPVJBJVTLMP
|
6.1 | Kd | 29 | — | |
UIARLYUEJFELEN
|
6.1 | Kd | 289 | Yes | |
PIMQWRZWLQKKBJ
|
6.1 | Kd | 36 | — | |
QQWUGDVOUVUTOY
|
6.1 | Kd | 231 | Yes | |
OYONTEXKYJZFHA
|
6.1 | Kd | 69 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |