Target Details
| UniProt AC | Q00536 |
|---|---|
| Gene Symbol | CDK16 |
| Protein Name | Cyclin-dependent kinase 16 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 73
- Clinical molecules 14
- Avg pChEMBL 7.32
Active Molecules (73)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GCIKSSRWRFVXBI
|
6.6 | Kd | 109 | Yes | |
XSDZPPRQLIZLDG
|
6.5 | IC50 | 6 | — | |
WVXNSAVVKYZVOE
|
6.5 | Kd | 92 | — | |
HMABYWSNWIZPAG
|
6.4 | IC50 | 12 | — | |
GRRYACDIYGRVLR
|
6.4 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
6.4 | Kd | 153 | — | |
PIQCTGMSNWUMAF
|
6.4 | Kd | 137 | Yes | |
BIIVYFLTOXDAOV
|
6.4 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
6.4 | Kd | 82 | Yes | |
HUXYBQXJVXOMKX
|
6.3 | Kd | 28 | — | |
ZNMYHQSTGGGHSX
|
6.3 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
6.2 | Kd | 231 | Yes | |
XWQVQSXLXAXOPJ
|
6.2 | IC50 | 7 | — | |
YYLKKYCXAOBSRM
|
6.1 | Kd | 191 | — | |
CXQHYVUVSFXTMY
|
6.0 | Kd | 154 | — | |
PSPFQEBFYXJZEV
|
6.0 | Kd | 10 | — | |
SEJGTFPOEJWEGG
|
6.0 | Kd | 149 | — | |
WBILCHGIPOEBGF
|
6.0 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
6.0 | Kd | 151 | — | |
BTIHMVBBUGXLCJ
|
6.0 | Kd | 21 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |