Target Details
| UniProt AC | Q00536 |
|---|---|
| Gene Symbol | CDK16 |
| Protein Name | Cyclin-dependent kinase 16 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 73
- Clinical molecules 14
- Avg pChEMBL 7.32
Active Molecules (73)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JRNJNYBQQYBCLE
|
9.3 | Kd | 40 | Yes | |
XXFHRRDNOYDSKG
|
9.1 | IC50 | 4 | — | |
NMXYXLBBQZYFDW
|
8.9 | IC50 | 4 | — | |
HGZJEOYIMBIRQI
|
8.7 | IC50 | 4 | — | |
OVPNQJVDAFNBDN
|
8.7 | Kd | 44 | Yes | |
NJIDANQIZWLYFH
|
8.6 | IC50 | 4 | — | |
XFCDYHLPKFWDMS
|
8.6 | IC50 | 4 | — | |
MANOLJFSBPUXMB
|
8.6 | IC50 | 4 | — | |
LXAGRPNIAUIQEA
|
8.6 | IC50 | 3 | — | |
TXUWSKNGSNTMNH
|
8.5 | IC50 | 2 | — | |
XLSYZSRXVVCHLS
|
8.5 | Kd | 48 | — | |
BQCPUBPCBQLKPP
|
8.5 | IC50 | 3 | — | |
IWFVOBVSODKUNF
|
8.3 | IC50 | 3 | — | |
OUSFTKFNBAZUKL
|
8.2 | Kd | 58 | Yes | |
JIBHJLIMQZDZRK
|
8.1 | IC50 | 3 | — | |
RMCYPGSJEZBAMX
|
8.1 | IC50 | 3 | — | |
NUPTZQFLDCQLOT
|
8.0 | IC50 | 4 | — | |
HZPYSAHDRSBARR
|
8.0 | IC50 | 4 | — | |
OQRVOQIHLQYVLO
|
8.0 | IC50 | 3 | — | |
FZWFQSYPXVHFDQ
|
8.0 | IC50 | 4 | — | |
AFFKASZZCVHEBW
|
7.9 | IC50 | 4 | — | |
RPGZQOOZHIEPJW
|
7.9 | Kd | 18 | — | |
RPGZQOOZHIEPJW
|
7.9 | Kd | 18 | — | |
BFSMGDJOXZAERB
|
7.9 | Kd | 33 | — | |
ODWIVHQPIGIBFU
|
7.9 | IC50 | 3 | — | |
INKWHXBJAUQYBV
|
7.8 | IC50 | 3 | — | |
PXQWBBNLJZQDEL
|
7.7 | IC50 | 4 | — | |
XZXHXSATPCNXJR
|
7.7 | Kd | 165 | Yes | |
KDKUVYLMPJIGKA
|
7.6 | Kd | 91 | Yes | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 213 | — | |
UIARLYUEJFELEN
|
7.6 | Kd | 289 | Yes | |
FLPXFWJMZVSLBP
|
7.5 | IC50 | 4 | — | |
LOLPPWBBNUVNQZ
|
7.5 | Kd | 97 | Yes | |
DKZYXHCYPUVGAF
|
7.5 | Kd | 112 | — | |
VXBAJLGYBMTJCY
|
7.5 | Kd | 34 | Yes | |
AXTAPYRUEKNRBA
|
7.4 | Kd | 24 | — | |
FGQPUEPSGPHCAO
|
7.3 | IC50 | 4 | — | |
UZWDCWONPYILKI
|
7.3 | Kd | 47 | — | |
RVKNONNXSNALJV
|
7.2 | IC50 | 21 | — | |
ZDQOAQIVXDLRDY
|
7.2 | IC50 | 4 | — | |
YKZGTZJVEPDXGU
|
7.1 | IC50 | 3 | — | |
GHOIKFWTAAALKT
|
7.0 | IC50 | 3 | — | |
RYCOMKGMIRGGDD
|
7.0 | IC50 | 4 | — | |
FLAQGMBHZVHXIW
|
6.9 | IC50 | 3 | — | |
KVPKTKLRKHRNNB
|
6.9 | IC50 | 2 | — | |
PIMQWRZWLQKKBJ
|
6.9 | Kd | 36 | — | |
PCHQRNIJFMRJNE
|
6.8 | IC50 | 4 | — | |
WINHZLLDWRZWRT
|
6.8 | Kd | 201 | Yes | |
KRIUNPBAQZGFQA
|
6.7 | Kd | 76 | — |