Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UAOIPNOTWOYAMU
|
7.2 | IC50 | 11 | Yes | |
XGWCLSYLELRSQN
|
7.2 | IC50 | 2 | — | |
ZHRBVPKKEHKSFH
|
7.2 | IC50 | 4 | — | |
HCRMONBJZIFRIR
|
7.2 | IC50 | 4 | — | |
LNLSVTCWVQLNIY
|
7.2 | IC50 | 2 | — | |
PBDNNWWYSHCMCH
|
7.2 | IC50 | 7 | — | |
WROPYEAREMSHKX
|
7.2 | IC50 | 2 | — | |
XVNXLMMYWHJXME
|
7.2 | IC50 | 2 | — | |
AKUJQCDZMJSNMC
|
7.2 | IC50 | 4 | — | |
BRQIEVOYMRUXNP
|
7.2 | IC50 | 7 | — | |
CFVOEIRDSYTLGT
|
7.2 | IC50 | 2 | — | |
GYEMABRPKRSBJU
|
7.2 | IC50 | 2 | — | |
SCACHXWSWJBIHG
|
7.2 | IC50 | 8 | — | |
SQUNOCMDMIQIQK
|
7.2 | IC50 | 10 | — | |
ULWKEYMEZWWCRY
|
7.2 | Ki | 5 | — | |
CXMKIWPGGSLHRE
|
7.2 | IC50 | 15 | — | |
KGLQVHSLHDKNTQ
|
7.2 | IC50 | 4 | — | |
XLUORARJPDKQIA
|
7.2 | IC50 | 3 | — | |
CIBYULXUPNERCM
|
7.1 | IC50 | 2 | — | |
NKSJUACUARPPLH
|
7.1 | IC50 | 13 | — | |
QIYYNXDEQKBHEH
|
7.1 | IC50 | 5 | — | |
SFDWUKJFXSWJPJ
|
7.1 | IC50 | 2 | — | |
WKEZGEHTYROLRA
|
7.1 | IC50 | 2 | — | |
KIHCZOJSOYPCCE
|
7.1 | IC50 | 2 | — | |
BEYPVZLSMWIZRD
|
7.1 | IC50 | 4 | — | |
JFEXQCAPNBAVHH
|
7.1 | IC50 | 2 | — | |
PMXCMJLOPOFPBT
|
7.1 | IC50 | 17 | Yes | |
ZPKXDHHDZZKMKI
|
7.1 | IC50 | 6 | — | |
JEWCMAYLACWOQD
|
7.1 | IC50 | 2 | — | |
YPSCKJWJIXZMSC
|
7.1 | IC50 | 15 | — | |
ZUCAWWSJZRVUAX
|
7.1 | Ki | 11 | — | |
AIQDZMUPVYDVLB
|
7.1 | Ki | 48 | — | |
BGNDQDYZQSRSAU
|
7.1 | IC50 | 3 | — | |
BGQVVTJSMBYUHC
|
7.1 | IC50 | 2 | — | |
GLDKGDSJAPIZTI
|
7.1 | IC50 | 2 | — | |
KVVMSGAISWJACO
|
7.1 | IC50 | 3 | — | |
LHQWPYOYDRVMFI
|
7.1 | Ki | 21 | — | |
LWANFAFTTOKZAX
|
7.1 | IC50 | 11 | — | |
LWANFAFTTOKZAX
|
7.1 | IC50 | 3 | — | |
MAUHUPWBMYAXPZ
|
7.1 | IC50 | 2 | — | |
QGFZDGFJYXGLAW
|
7.1 | IC50 | 3 | — | |
QQWUGDVOUVUTOY
|
7.1 | Ki | 231 | Yes | |
UIRCQOKSJDLYBB
|
7.1 | Ki | 50 | — | |
WYEXOAKSTKXOBU
|
7.1 | IC50 | 3 | — | |
YMIJUBCSOKSFRU
|
7.1 | Ki | 87 | — | |
DDLZLOKCJHBUHD
|
7.1 | IC50 | 23 | — | |
HGRMYMRCAGWXEQ
|
7.1 | IC50 | 6 | — | |
HKSZLNNOFSGOKW
|
7.1 | Kd | 213 | — | |
OLOJSTRISMGUEK
|
7.1 | IC50 | 5 | — | |
PFDVIMSWMQLRQB
|
7.1 | IC50 | 2 | — |