Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IPSJLLWTAZLENF
|
7.3 | IC50 | 2 | — | |
RXGOWNXDRJHZDW
|
7.3 | IC50 | 2 | — | |
DPFVGQNGSOMJSY
|
7.3 | IC50 | 2 | — | |
JLKHGQLTVZHANW
|
7.3 | IC50 | 2 | — | |
VCEUNJCUQFBRBD
|
7.3 | IC50 | 2 | — | |
CQGFDYLOZSKCBQ
|
7.3 | IC50 | 2 | — | |
KDKUVYLMPJIGKA
|
7.3 | Kd | 91 | Yes | |
LQHMJVOJVOLFTJ
|
7.3 | IC50 | 7 | — | |
PUXKEKPYASIYGT
|
7.3 | IC50 | 7 | — | |
ZJKDYTFNXUBLEQ
|
7.3 | IC50 | 15 | — | |
ZITKTAJHKVYGTC
|
7.2 | IC50 | 7 | — | |
HONCRTYDCHPQOK
|
7.2 | IC50 | 2 | — | |
WRPCQNMNBWSPBJ
|
7.2 | IC50 | 2 | — | |
XNKBKFNLOYVTSF
|
7.2 | IC50 | 11 | — | |
AYSFEKIVJXIJTM
|
7.2 | IC50 | 8 | — | |
BOPIEFLHGAQWGB
|
7.2 | IC50 | 3 | — | |
HLSGDZZAUXGGFJ
|
7.2 | Ki | 4 | — | |
LQYHWFFRRIMAPW
|
7.2 | IC50 | 2 | — | |
RSPXQCXRWMXEAA
|
7.2 | IC50 | 2 | — | |
SBNNOXYSSSCMJX
|
7.2 | IC50 | 6 | — | |
SJJOSGWHLXBKSU
|
7.2 | IC50 | 2 | — | |
TUMYZJPVQGGVEN
|
7.2 | IC50 | 7 | — | |
GRMBHDGZBLMPSZ
|
7.2 | IC50 | 2 | — | |
JBTRAENEEJNXFX
|
7.2 | IC50 | 2 | — | |
KCGZOQMFGRRYKH
|
7.2 | IC50 | 3 | — | |
KKNOSXFGCMVMNP
|
7.2 | IC50 | 2 | — | |
MAIBFWJHQLEUMH
|
7.2 | IC50 | 2 | — | |
NGFGTMFVWSDFPS
|
7.2 | IC50 | 32 | — | |
WMIYIBXBFBOKCT
|
7.2 | IC50 | 6 | — | |
YOOLJWCJXSFKSE
|
7.2 | IC50 | 2 | — | |
BKBCSMDCCAWWNC
|
7.2 | Ki | 7 | — | |
BQWACEUCYSZDBQ
|
7.2 | Ki | 5 | — | |
CYLGCMABIBXHIQ
|
7.2 | Ki | 16 | — | |
HQUWRDCCNSLORW
|
7.2 | IC50 | 2 | — | |
KTWBYGUSEYSRND
|
7.2 | Ki | 28 | — | |
LCHCSKHPVCDXAU
|
7.2 | Ki | 30 | — | |
MHWHPWMWKYXCRJ
|
7.2 | Ki | 32 | — | |
PCQMERRARZKTPW
|
7.2 | Ki | 68 | — | |
RFBPWKMQWSIPEO
|
7.2 | Ki | 28 | — | |
RRAMBEGOYIJQHY
|
7.2 | Ki | 11 | — | |
UMTWTCVTRDYHQQ
|
7.2 | Ki | 56 | — | |
YWTBGJGMTBHQTM
|
7.2 | Ki | 65 | — | |
FRLPUUILIGCJSG
|
7.2 | IC50 | 2 | — | |
IGRZXNLKVUEFDM
|
7.2 | IC50 | 8 | — | |
IHBOEHLUIBMBMY
|
7.2 | IC50 | 7 | Yes | |
MOFKVWKHBJPHSX
|
7.2 | IC50 | 2 | — | |
NUBBIJVOSXWZTF
|
7.2 | IC50 | 13 | — | |
QQXOHTCNPILOGG
|
7.2 | IC50 | 3 | — | |
QYCAOWUXVAQWNK
|
7.2 | IC50 | 2 | — | |
SHHLIGVBIWQSRR
|
7.2 | IC50 | 4 | — |