Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RGNHKJWHFIPHIM
|
7.4 | Ki | 66 | — | |
RMEWJCSHDSUJKS
|
7.4 | IC50 | 2 | — | |
DHPKYHMTJHTQKB
|
7.4 | IC50 | 2 | — | |
HFEVNTGRPXCJIM
|
7.4 | IC50 | 6 | — | |
LIJUCWLALFXGCL
|
7.4 | IC50 | 7 | — | |
PGVAPFNXIBFQNO
|
7.4 | IC50 | 3 | — | |
UVMVCEDKKHGTIW
|
7.4 | IC50 | 7 | — | |
CNNQBAXDFGTALM
|
7.4 | IC50 | 5 | — | |
GPSDJCPWZFYLRU
|
7.4 | IC50 | 2 | — | |
QYNVMKNYPFKRBL
|
7.4 | Ki | 9 | — | |
QZTJCAGUOSLOOZ
|
7.4 | IC50 | 2 | — | |
SBNNOXYSSSCMJX
|
7.4 | IC50 | 6 | — | |
UUFIEDRPFIIXAY
|
7.4 | Ki | 6 | — | |
ZPKXDHHDZZKMKI
|
7.4 | IC50 | 6 | — | |
ANELMUPUYRZVHZ
|
7.4 | IC50 | 7 | — | |
BHGNYQXAUNNTRE
|
7.4 | IC50 | 2 | — | |
OSZOLMOXJMNVGS
|
7.4 | IC50 | 4 | — | |
BNARYBDTYNEVER
|
7.4 | IC50 | 3 | — | |
CJLTWANHPMOFEB
|
7.4 | IC50 | 3 | — | |
FEUVVQAFOCJYBF
|
7.4 | IC50 | 2 | — | |
JVLUKLANRWXEHV
|
7.4 | IC50 | 2 | — | |
KEUUTBKQXWXFLI
|
7.4 | IC50 | 5 | — | |
LBVIZFWUIQSZHP
|
7.4 | IC50 | 10 | — | |
MJMQYAHYXBAAPB
|
7.4 | IC50 | 3 | — | |
URMALQKFRQFSGH
|
7.4 | IC50 | 2 | — | |
CQZDWCOZFXQUFP
|
7.3 | IC50 | 2 | — | |
DBDLWYCQSVIKRY
|
7.3 | IC50 | 2 | — | |
KAMWROHYXYCDLF
|
7.3 | IC50 | 2 | — | |
IRLVKSQKZPUCOP
|
7.3 | IC50 | 2 | — | |
RLVCFRZZHAKDOE
|
7.3 | IC50 | 6 | — | |
IHKXIGRVBUPRKQ
|
7.3 | IC50 | 3 | — | |
LBPVERPKZZCMIU
|
7.3 | IC50 | 2 | — | |
NGLJEWVPKWMIAJ
|
7.3 | IC50 | 5 | — | |
SMWJYKRUKGMKJV
|
7.3 | IC50 | 11 | — | |
ULNGKSGQVVQHJF
|
7.3 | IC50 | 2 | — | |
GVIGDUKISNSSHK
|
7.3 | IC50 | 3 | — | |
AWJPVXSHMIELNJ
|
7.3 | Ki | 23 | — | |
FSEJNURQBJZNAM
|
7.3 | IC50 | 2 | — | |
JYGNOLIKBUTZNC
|
7.3 | IC50 | 8 | Yes | |
LBVKEEFIPBQIMD
|
7.3 | Ki | 27 | — | |
NTHMDBBWWNTVAZ
|
7.3 | IC50 | 5 | — | |
PJROIFLISSJQQQ
|
7.3 | IC50 | 4 | — | |
PRJNNPMIUGYOST
|
7.3 | IC50 | 14 | — | |
RAFWSIQGGUBJOQ
|
7.3 | IC50 | 2 | — | |
SVBJNUDKKXGVHI
|
7.3 | IC50 | 6 | — | |
WROPYEAREMSHKX
|
7.3 | IC50 | 2 | — | |
XPHWIERLJBFPFV
|
7.3 | Ki | 69 | — | |
YEHCNYAQEBQCCS
|
7.3 | Ki | 74 | — | |
YXUQWISLOFXNGN
|
7.3 | Ki | 16 | — | |
GNTSKAUZBDGNGK
|
7.3 | IC50 | 6 | — |