Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MKNYSPZGSGBELV
|
7.5 | IC50 | 2 | — | |
NSEKTECTEUZVNV
|
7.5 | IC50 | 4 | — | |
PHZDWQYTFQOSSZ
|
7.5 | IC50 | 15 | — | |
SLKSRHOPMDATBX
|
7.5 | IC50 | 5 | — | |
UBLFSMURWWWWMH
|
7.5 | IC50 | 7 | — | |
UEFVCKVWJQJSDH
|
7.5 | IC50 | 2 | — | |
XHJMMMPXTUEBMQ
|
7.5 | IC50 | 4 | — | |
JFHNULPYENHDTR
|
7.5 | IC50 | 2 | — | |
TVQIAQPBIDLYOL
|
7.5 | IC50 | 4 | — | |
ZOPGCNRZFZPRGB
|
7.5 | Ki | 9 | — | |
CNQGNADBGYCKKV
|
7.5 | Ki | 25 | — | |
OYPIIVNTYVSCNV
|
7.5 | IC50 | 4 | — | |
QLWUDWMYFSWGHK
|
7.5 | Ki | 22 | — | |
RWKDVIAVTRRJIR
|
7.5 | Ki | 23 | — | |
VGGPBVXGHSIMPS
|
7.5 | IC50 | 4 | — | |
VTQQYBGURNVVFE
|
7.5 | Ki | 17 | — | |
XNWKXXIGSPPPBH
|
7.5 | Ki | 31 | — | |
YWITWZUKNXWOSD
|
7.5 | Ki | 10 | — | |
KVZRUJJMBHTJLY
|
7.5 | IC50 | 2 | — | |
PPSLREGORUQEEL
|
7.5 | IC50 | 2 | — | |
SHBOZSJPVRMXBA
|
7.5 | IC50 | 7 | — | |
SPKWRLBKVPRPMT
|
7.5 | IC50 | 9 | — | |
TVARIYLSKVWCHN
|
7.5 | Ki | 11 | — | |
DBKUHLGRJZFKQS
|
7.5 | IC50 | 5 | — | |
FULPDCCIDPUWGS
|
7.5 | IC50 | 4 | — | |
GNHNRVSQWNAGHC
|
7.5 | IC50 | 7 | Yes | |
KGMVZSJAPXYTKH
|
7.5 | IC50 | 23 | — | |
LNGGMJFRIWMXLS
|
7.5 | IC50 | 2 | — | |
FDJQQPZQIBTWLE
|
7.5 | IC50 | 4 | — | |
PWWHQERJKXLERO
|
7.5 | IC50 | 2 | — | |
LLFOBMRPWNABCB
|
7.5 | IC50 | 11 | — | |
BUVUGYVWVBFUMI
|
7.4 | Ki | 11 | — | |
BYFFLCLXJMXMTM
|
7.4 | IC50 | 2 | — | |
FJINXQDJHXTMEL
|
7.4 | Ki | 9 | — | |
DSMBDRWDECFDNR
|
7.4 | IC50 | 7 | — | |
FYBVVRIGUJAAOT
|
7.4 | IC50 | 2 | — | |
JESHQJYUKOEMIP
|
7.4 | IC50 | 3 | — | |
QNUKRWAIZMBVCU
|
7.4 | IC50 | 17 | Yes | |
RPYUTGQONYNCSI
|
7.4 | IC50 | 4 | — | |
VDTYYNPPVROBPA
|
7.4 | IC50 | 4 | — | |
FQFGDUPFMGYOMB
|
7.4 | IC50 | 6 | — | |
HCEVZIBGQRWFCG
|
7.4 | IC50 | 9 | — | |
HEPOPUWWRFFLLL
|
7.4 | IC50 | 2 | — | |
KMWYBWMCMDBJGT
|
7.4 | IC50 | 2 | — | |
PDAAWAZSKXRPAS
|
7.4 | IC50 | 2 | — | |
DWDSNANBEINKNN
|
7.4 | IC50 | 4 | — | |
BIDYUGXUCHBVIV
|
7.4 | IC50 | 2 | — | |
HKOGEZCYHMAXBA
|
7.4 | IC50 | 2 | — | |
OLUKILHGKRVDCT
|
7.4 | IC50 | 44 | Yes | |
PJUVRETYCLPAFV
|
7.4 | Ki | 20 | — |